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N-(3,4-dimethylphenyl)-4-(pyridin-3-yloxy)piperidine-1-carboxamide
5-{3-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]propyl}-1,3,4-thiadiazol-2-amine
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]propanamide
4-benzoyl-6-(benzyloxy)-1-(2-methylpropyl)-1,4-diazepan-2-one
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-4-(1H-pyrazol-1-yl)butan-1-one
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-{2-[4-(2-cyclohexylacetyl)piperazin-1-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(1,3-dihydro-2-benzofuran-5-yl)urea
(4aS,8aR)-1-(3-aminopropyl)-6-[(3-methyl-1,2-benzoxazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
6-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]quinoxaline
[(3R,4R)-1-(1H-1,3-benzodiazole-5-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(4-{[1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-(2-hydroxyethyl)-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
2-cyclopentyl-8-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
3-hydroxy-3-{[(2-methoxyethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-ethyl-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(1-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)phenol
[(3-methoxyphenyl)methyl](prop-2-en-1-yl)(quinoxalin-2-ylmethyl)amine
(1S,9S)-11-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(piperidin-1-yl)butan-1-one
4-(3-chloro-5-fluorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
5-acetyl-N-{[2-(trifluoromethyl)phenyl]methyl}thiophene-3-carboxamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
1-(2,5-dimethylfuran-3-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N,N-dimethyl-5-{[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]methyl}furan-2-carboxamide
N-[1-(furan-2-yl)ethyl]-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
(1-methyl-1H-imidazol-2-yl)(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)methanol
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}propanamide
(3E)-1-[1-(hydroxymethyl)-9-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]hex-3-en-1-one
1-[(4-fluorophenyl)methyl]-4-[(quinoxalin-2-yl)amino]pyrrolidin-2-one
N3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
5-{[4-(5-methylfuran-2-yl)phenyl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-(2H-1,2,3-benzotriazol-2-yl)-1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}ethan-1-one
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dihydro-1-benzofuran-5-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]thiophene-3-carboxamide
1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-[7-(furan-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-3-methoxypiperidine
3-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-methyl-1-[4-methyl-3-(propan-2-yl)phenyl]urea
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-ethylpyrimidin-2-amine
1-(4-cyano-2-fluorophenyl)-3-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}urea
8-(2-oxoimidazolidine-4-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(2,3-dihydro-1H-inden-2-yl)-4-(furan-3-carbonyl)-1,4-diazepane
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(pyrimidin-4-ylmethyl)amine
1-[2-(dimethylamino)-4-{[2-(morpholin-4-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-cyclopropyl-N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
{1-[(2,5-dimethylfuran-3-yl)methyl]piperidin-2-yl}methanol
2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1-methyl-1H-indole