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4,4-difluoro-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
2-[5-(6-methyl-2-propylpyrimidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(4-fluorophenyl)methyl]piperidine-4-carboxamide
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(4-ethoxy-2-fluorophenyl)urea
4-[(2-aminopyridin-3-yl)methyl]-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(4,6-dimethylpyrimidin-2-yl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4R)-3-hydroxy-1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]piperidin-4-yl]pyridine-2-carboxamide
N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-phenyl-1,2-oxazole-5-carboxamide
2-[5-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
methyl 6-[1-(4-fluorophenyl)propan-2-yl]-2-[(2-methoxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-4-methyl-N-(pyridin-3-ylmethyl)benzamide
5-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-(2H-indazol-2-yl)ethan-1-one
(2S,4R)-4-amino-1-(2,2-dimethylpent-4-en-1-yl)-N,N-diethylpyrrolidine-2-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
N-[1-(2-phenylethyl)piperidin-3-yl]-2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetamide
(3aR,6aR)-2-ethyl-5-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclohex-3-ene-1-carboxamide
5-(1-cyclopentyl-1H-imidazol-2-yl)-2-(furan-2-yl)pyrimidine
5-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-methyl-3-({8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1,2-dihydroquinolin-2-one
1-(3,4-dimethoxyphenyl)-2-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-amine
N-[4-(difluoromethoxy)-2-methylphenyl]-4-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
(4S)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-bromobenzamide
N-cyclohexyl-3-{[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]amino}propanamide
N-(cyclohexylmethyl)-2-cyclopropyl-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(4-methylphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-acetyl-N-[2-(3-methylthiophen-2-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{5-[1-(furan-2-ylmethyl)piperidin-4-yl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}pyridine
N-cyclopropyl-1,6-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-(propan-2-yl)pyrimidin-4-amine
1-(3,6-dimethylpyrazin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
N-{[4-hydroxy-1-(2-methylfuran-3-carbonyl)azepan-4-yl]methyl}morpholine-4-carboxamide
9-[3-(1H-imidazol-1-yl)propyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-[(3R,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(4aS,8aR)-6-(1H-1,3-benzodiazol-2-ylmethyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
(1R,5R)-3-[2-(2-ethoxyethoxy)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-{[1-(methoxymethyl)cyclopentyl]methyl}-1-(quinolin-5-yl)urea
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-ethylpyridine-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
(3R,4R)-1-(5-fluoropyrimidin-2-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-methyl-8-[3-(2-methylphenyl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(5S)-5-{3-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
2-{1-[(3-methoxyphenyl)methyl]-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(pyrimidin-4-ylmethyl)benzamide
(3R)-N-[4-chloro-3-(furan-2-amido)phenyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide