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1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-fluorophenyl)propan-1-one
1-(2-benzylmorpholin-4-yl)-4-phenylbutane-1,2-dione
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-3-yl)piperazine
N-(2H-1,3-benzodioxol-4-ylmethyl)-4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
N-(3,5-dimethylphenyl)-2-oxo-2-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]acetamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(3-methylthiophen-2-yl)methyl]benzamide
N-{2-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
1-(3,4-dimethylphenyl)-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-3-(2-methylpropyl)-1H-1,2,4-triazole
6-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
2-{[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
4-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}butan-1-ol
4-{[2-(2-chlorophenoxy)ethyl]amino}-2-methylpentan-2-ol
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N,2,2-trimethyl-4-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3,4-dihydro-2H-pyran-6-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
2-benzyl-9-(5-methylpyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}benzamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(thiophen-3-yl)acetamide
N-(furan-3-ylmethyl)-4-[(oxolan-2-ylmethyl)sulfamoyl]benzamide
ethyl({2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}sulfamoyl)methylamine
8-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(2-fluorophenyl)piperidin-4-yl]-3-(piperidin-3-yl)benzamide
1'-{[5-(4-chlorophenyl)furan-2-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 4-(5-{[methyl(thiophen-3-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
(3R,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-indole-3-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-1,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-1,3-thiazol-4-yl}methanol
1-methyl-2-{1-[(3,4,5-trimethoxyphenyl)methyl]-1H-imidazol-2-yl}-1H-imidazole
3-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(4-methanesulfonylphenyl)urea
3-benzyl-1-methyl-3-[2-oxo-2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-indol-2-one
2-(morpholin-3-yl)-1-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
[(2S,6S)-4-[(2,3-difluorophenyl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(furan-2-yl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(3-methylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-benzoyl-1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
1-[(2,4-dimethoxyphenyl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-phenoxypropyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-5-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidine
9-[(5-ethylfuran-2-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2,6-dimethoxyphenyl)-5-methyl-1H-indazole
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
4-[(1S,2S)-2-hydroxycyclohexyl]-N-[3-(trifluoromethyl)phenyl]piperazine-1-carboxamide
N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-1-(propan-2-yl)-1H-pyrazole-5-carboxamide
6-(hydroxymethyl)-N-(3-methylcinnolin-5-yl)-1,4-oxazepane-4-carboxamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
N-cyclohexyl-3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}propanamide
(3S)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
(2S,4S)-1-cyclopentyl-N-ethyl-4-[3-(2-fluorophenyl)propanamido]pyrrolidine-2-carboxamide