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2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methoxyphenyl)ethyl]acetamide
6,7-difluoro-3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
2-(dimethylamino)-2-(4-methylphenyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N-(propan-2-yl)pyrimidin-4-amine
N-[(4-hydroxyazepan-4-yl)methyl]-4-(2-methoxyphenyl)benzamide
1-(1-cyclopentyl-1H-pyrazol-5-yl)-3-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]urea
[1-cyclohexyl-3-(3-methoxypropyl)piperidin-3-yl]methanol
1-{2-[(2-methyl-1-benzofuran-5-yl)formamido]ethyl}piperidine-3-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
N-benzyl-N-ethyl-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(3,5-difluorophenyl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(6-cyanopyridin-3-yl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
1-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propan-2-ol
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,4-triazol-3-amine
3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
2-(4-chloro-2-{[ethyl(oxan-2-ylmethyl)amino]methyl}phenoxy)acetic acid
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-methyl-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-methyl-N-(1-methylpiperidin-4-yl)-3-[1-(5-phenylpentanoyl)piperidin-3-yl]propanamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-[(6-chloro-2-fluoro-3-methoxyphenyl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-amino-6-{2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-2-(1H-pyrazol-1-yl)butanamide
2-[5-(2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-6-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
2-methyl-3-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]-N-(1,3-thiazol-2-yl)benzamide
(3R,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
methyl 4-(5-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
6-chloro-N-(oxan-3-yl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
2-[1-(quinoline-8-carbonyl)pyrrolidin-3-yl]benzoic acid
2-butyl-5-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzoxazole
2-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methylpyrazine
1-(4-fluorophenyl)-4-[1-(naphthalene-2-carbonyl)piperidin-3-yl]piperazine
2-({6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidin-3-yl}formamido)-N,N-dimethylpropanamide
N-benzyl-5-[1-(5-methylpyridin-3-yl)-1H-imidazol-2-yl]pyrimidin-2-amine
(3S,4R)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
(1S,5R)-3-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-chloro-4-fluorophenoxymethyl)-N,N-diethyl-1,3-oxazole-4-carboxamide
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-4-({[(2-methoxyphenyl)methyl]amino}methyl)-2-methylpyrrolidin-2-yl]methanol
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepane
2-{4-[4-(2,3-dihydro-1H-isoindole-2-carbonyl)-8-methylquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
2-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
ethyl 2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}-1,3-oxazole-4-carboxylate
(3R)-3,4,4-trimethyl-1-[1-methyl-5-(trifluoromethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carboxylic acid
(1R,3S)-3-(2-aminoethoxy)-7-[(5-phenylthiophen-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol