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N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-3-propyl-1H-pyrazole-5-carboxamide
(3E)-1-[3-(3,4-dichlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pent-3-en-1-one
N,N-dimethyl-4-(3-phenylpiperazine-1-carbonyl)piperidine-1-carboxamide
5-[2-({[1-(2,2-dimethylpropyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-6-hydroxy-1,4-diazepan-1-yl)-2-methoxyethan-1-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-methyl-1H-pyrrole-3-carboxamide
5-(2,6-difluoro-4-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-{5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(morpholin-4-yl)propan-1-one
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)cyclohexanecarboxamide
[1-(2-fluorobenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
2-(azepan-1-yl)-1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]acetamide
3-methyl-7-(4-methylpyrimidin-2-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(4aS,8aR)-6-[(3-hydroxyphenyl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-cyclohexylpiperidine-3-carboxamide
(2R,6R)-4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-(3-hydroxy-3-methylbutyl)-N-[2-(pyridin-4-yl)ethyl]benzamide
1-(1-methyl-1H-pyrazole-5-carbonyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
6-(benzyloxy)-4-(2,3-dihydroxypropyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
8-fluoro-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
(2S,4S)-4-amino-N-[(3-methoxy-2-propoxyphenyl)methyl]-1-methylpyrrolidine-2-carboxamide
(2E)-3-(2-chlorophenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}prop-2-enamide
(1R,5S,8R)-3-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-azabicyclo[3.2.1]octan-8-ol
3-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1λ6-thiolane-1,1-dione
3-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-2,8-diazaspiro[4.5]decane
3-methyl-7-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(1S,5R)-3-(oxan-4-yl)-6-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
6-[4-(4-chlorophenoxy)piperidin-1-yl]pyridine-2-carboxylic acid
6-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanamide
4-({[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-methoxyphenol
(4aR,8aR)-2-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-(1-benzylpiperidin-3-yl)-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
benzyl 3-(3-methoxy-5-methylthiophene-2-amido)pyrrolidine-1-carboxylate
5-{2H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-(2-{[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-{[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]methyl}-6-fluoroquinolin-4-ol
6-cyclopentyl-1-methyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3aR,7aS)-2-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-1,4-diazepan-2-one
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N1-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]piperidine-1,3-dicarboxamide
3-(1H-indol-2-ylmethyl)-3,9-diazaspiro[5.5]undecane
1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(pyrrolidine-1-carbonyl)piperidine
2-methoxy-N-methyl-5-({methyl[3-(3-methylphenoxy)propyl]carbamoyl}amino)benzamide
3-(4-methoxy-2-methylbenzoyl)-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidine
2-methyl-4-(1,4-oxazepan-4-ylmethyl)quinoline
N-(2-chloropyridin-3-yl)-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide