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8-methyl-5-[2-(piperazin-1-yl)phenyl]quinoline
[4-({1-[3-(dimethylamino)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
(2R,3R)-3-[(3-methoxypropyl)(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(1-butylpiperidin-4-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
3-(pentan-2-yl)-8-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N,N-diethylpiperidine-4-carboxamide
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-(oxan-3-ylmethyl)-3-sulfamoylbenzamide
2-{[2-(hydroxymethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-benzyl-N-ethyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,2R)-2-({[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)cyclohexan-1-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}propanamide
5-{2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}pyrrolidin-2-one
3-[({1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
4-(5-propylpyrimidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
10-methoxy-5-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-(methoxymethyl)-N-methyl-N-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]cyclopropan-1-amine
methyl (2S)-1-(5-benzenesulfonamido-1-ethyl-2-methyl-1H-1,3-benzodiazole-7-carbonyl)pyrrolidine-2-carboxylate
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
(2S)-N-(3-methanesulfonamido-4-methoxyphenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
4-{[2-(2-fluorophenyl)ethyl]amino}-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
[7-(3,5-dimethyl-1H-pyrazol-4-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-(quinoxalin-2-ylmethyl)acetamide
3-(2-methoxyphenyl)-6-(4-methylthiophen-3-yl)pyridazine
N-(1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
N-(carbamoylmethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-({[2-(azepan-1-yl)ethyl](methyl)amino}methyl)benzoic acid
N-cycloheptyl-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
6-(benzyloxy)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
2-(2,4-dichlorophenyl)-4-methoxypyrimidine
(3aS,6aS)-2-cyclohexyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-(cyclohexylmethyl)-2-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-N,N-diethyl-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N,2-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]imidazo[1,2-a]pyrimidine-3-carboxamide
N-[2-(3-fluorophenyl)ethyl]-2-(1H-imidazol-2-yl)benzamide
1-[(1R,5R)-6-[(2,4-diethoxy-3-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
4-methyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-(2-fluorophenoxymethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
N,1-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
1-methanesulfonyl-N-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidin-4-amine
2-(3-cyano-3,3-diphenylpropyl)benzene-1-sulfonamide
3-[3-(dimethylamino)phenyl]-1-(3-hydroxypropyl)-1-(pyridin-3-ylmethyl)urea
6-(5-ethoxy-2-methyl-1-benzofuran-3-carbonyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
8-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzenesulfonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{[1-(6-methoxypyridin-2-yl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(3-ethoxy-4-methoxyphenyl)methyl]-N-methylacetamide
5-fluoro-2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole