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2-(2-methanesulfonylacetyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-methyl-3-phenyl-8-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,8-diazaspiro[4.5]decan-2-one
(3R,4S)-4-{[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](ethyl)amino}oxolan-3-ol
2,6,8-trimethyl-4-(thiomorpholine-4-carbonyl)quinoline
3-[2-(methylamino)ethyl]-1-[2-(prop-2-en-1-yloxy)phenyl]urea
2-ethoxy-5-{2-[(3R)-3-hydroxypyrrolidin-1-yl]pyrimidin-4-yl}benzoic acid
N-[cyclohexyl(thiophen-2-yl)methyl]-1-methylpiperidin-4-amine
[(3R,4S)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-(7-hydroxy-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
2-(2-aminoethyl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]quinazolin-4-amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]benzamide
3-(3-chlorobenzoyl)-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}piperidine
4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1-(3,5-dimethylphenyl)piperazin-2-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
1'-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(1-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1-hydroxy-2-methylpropan-2-yl)propanamide
{5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]furan-2-yl}methanol
2-[(3,4-difluorophenyl)methyl]-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(2,3-dihydro-1-benzofuran-2-ylmethyl)({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
8-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidine
7-[(2,3-difluorophenyl)methyl]-2-(3,5-dimethylfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
2-{[(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
8-(4-methanesulfonylphenyl)-1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
1-methyl-1'-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-{5-methyl-4-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
1-(4-aminopyrimidin-2-yl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-methylacetamide
2-(2-fluoro-4-methylphenyl)-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}acetic acid
(4aR,7aS)-N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(azepan-2-ylmethyl)-3-(2,5-difluorophenyl)urea
1-(5-fluoropyrimidin-2-yl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-(5-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
3-{[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(trifluoromethyl)pyridine
2-[1-(cyclohexylmethyl)-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N4-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidine-4,6-diamine
4-(furan-2-ylmethyl)-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperazine-2-carboxylic acid
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(furan-3-ylmethyl)methylamine
(1R,5R)-3-methanesulfonyl-N-(thiophen-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(1S,6R)-3-methyl-9-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(3R,4S)-1-(furan-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2-(2-methoxyethyl)piperidine
(1S,5R)-6-(5-fluoro-2-methylbenzoyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3,4-difluorophenyl)methyl]-3-[1-(furan-3-carbonyl)piperidin-3-yl]propanamide
N-(2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethyl)-1,3-thiazole-5-carboxamide