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N-{3-[(4-methylphenyl)sulfanyl]propyl}-3-(2-oxoimidazolidin-1-yl)benzamide
1,3-dimethyl-5-{2-[3-(2-methylphenoxy)azetidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
methyl (1S,3S,3aR,6aS)-3-(2-chloro-6-fluoro-3-methoxyphenyl)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-methyl-1,3-thiazole-4-carboxamide
N-benzyl-N-methyl-3-[1-(2-phenoxyacetyl)piperidin-4-yl]propanamide
(3S,4S)-1-[(2E)-2-methylbut-2-en-1-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
N-methyl-5-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
{1-[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
[(3R,4R)-1-(3-ethyl-1H-indole-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[2-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)ethyl]-1,2-dihydropyridin-2-one
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-(5-methylthiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(azepan-1-yl)propyl]-N-methyl-2-[(prop-2-en-1-yl)amino]benzamide
N-{[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-3-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
(3R,4R)-1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
(3S,4S)-4-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-ol
2-(2-hydroxypropyl)-9-(3-methylthiophene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-(2-methylpropyl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-({1-[(1-hexylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)azetidin-3-ol
7-methyl-2-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
1-(4-carbamoyl-1,3-thiazol-2-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(1S,5R)-3-benzyl-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carbonyl}-N,N-dimethylpiperazine-1-sulfonamide
2-(1H-imidazol-2-yl)-N-[2-(pyridin-3-yl)ethyl]benzamide
7,7-dimethyl-2-(2-propoxyethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[cyclopentyl(methyl)amino]-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
4-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-4H-1,2,4-triazole
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(trifluoromethyl)piperidine
5-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
2-[1-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-4-yl]-N,N,6-trimethylquinoline-4-carboxamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)(2-phenylethyl)amine
N-[(3S,4R)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(3-methoxyphenyl)-1-[2-(pent-4-enamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-({[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]carbamoyl}amino)-N,N,2-trimethylbenzamide
2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-ol
9-ethyl-N-(5-fluoro-2-methylphenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
4-(8-chloroquinolin-2-yl)-1-[(3,4-dimethylphenyl)methyl]piperazin-2-one
2-{4-[(2E)-3-phenylprop-2-en-1-yl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]butan-1-one
N-ethyl-N-methyl-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
1-(2-{[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
2-(2-methyl-1,3-thiazol-4-yl)-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}acetamide
1-(6-{methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
1-[2-methyl-7-(6-methylpyridazin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-ol
4-methoxy-2-({4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)pyridine
[(5-ethylpyridin-2-yl)methyl](methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
N-[3-(methylsulfanyl)phenyl]-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
1-ethyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide