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(2S,4R)-4-amino-N-methyl-1-(9H-purin-6-yl)pyrrolidine-2-carboxamide
N-({5-[(2,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
5-(1H-imidazol-1-ylmethyl)-N-(isoquinolin-5-ylmethyl)-N-methylpyridin-2-amine
3-acetyl-N-[1-(3,4-dimethoxyphenyl)propyl]-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-(oxan-4-yl)-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,N-bis(1,3-oxazol-4-ylmethyl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-(1H-pyrrol-1-yl)pentan-1-one
1-ethyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
2-(1H-imidazol-4-yl)-4,5,6,7-tetramethyl-1H-1,3-benzodiazole
2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-8-(1-methoxypropan-2-yl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-{4-[2-amino-3-cyano-6-(thiophen-2-yl)pyridin-4-yl]-1H-pyrazol-1-yl}propanoate
N-[2-(dimethylamino)ethyl]-4-fluoro-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)benzamide
1-[2-(morpholin-4-yl)ethyl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-{[6-(methoxymethyl)pyrimidin-4-yl](methyl)amino}-1-phenylpropan-1-ol
2-[benzyl(methyl)amino]-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(3S,4S)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamide
2-{9-[(2,3-difluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
5-methoxy-1-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-indole-2-carboxamide
4-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-2,3-dihydro-1H-inden-1-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
9-ethyl-N-(3-methoxyphenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-methyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
5-[5-(diethylcarbamoyl)furan-2-yl]thiophene-2-carboxylic acid
1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-[2-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(2R)-2-hydroxy-1-[4-(3-methylphenoxy)piperidin-1-yl]-2-phenylethan-1-one
1-({2-[3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)piperidine-3-carbonitrile
N-(2H-1,3-benzodioxol-5-yl)-1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}piperidin-3-amine
5-(4-methoxyphenyl)-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,2,4-triazin-3-amine
1-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-4-yl}piperidin-3-ol
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(3-chlorophenyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
2-(dimethylamino)-N-[(5-ethylpyridin-2-yl)methyl]-2-(2-methylphenyl)acetamide
(3S)-N,N-dimethyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}azepan-3-amine
N-ethyl-5-methoxy-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-2-carboxamide
2-({[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}amino)pyridine-4-carboxamide
1-(4-methoxy-2-methylphenyl)-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
(4aS,7aR)-1-cycloheptanecarbonyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-1-(2-methyl-1,3-benzoxazole-6-carbonyl)-1,4-diazepan-5-one
3-{[7-(hydroxymethyl)-9-[3-(methylsulfanyl)propyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl}phenol
1-(cyclopropylmethyl)-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}thiomorpholine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(2-methoxyacetyl)piperidine-3-carboxamide
{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
dimethyl({[4-methyl-5-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine