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N-(2,3-dimethylphenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{8-[4-(difluoromethoxy)benzoyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
5-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
3-methyl-8-[(1-propyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-5-methoxy-3-methyl-1H-indole
2-{4-[(3,5-difluorophenyl)methyl]piperazine-1-carbonyl}-5-methoxy-1,4-dihydropyridin-4-one
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
[1-(3-methylthiophene-2-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
6-ethoxy-2-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}quinoline
1-(ethanesulfonyl)-3-[2-(3-fluorophenyl)ethyl]piperidine
N-[(2-fluorophenyl)methyl]-3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}propanamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
1-[(4aR,8aR)-7-(3-chloro-2-methylbenzoyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-[(3-methyloxetan-3-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
4-methoxy-2-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyrimidine
(1R,2S)-N-butyl-2-[3-(pyridin-3-yl)azetidine-1-carbonyl]cyclohexane-1-carboxamide
4-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1λ6-thiomorpholine-1,1-dione
N-(diphenylmethyl)-2-{[(1R,4S)-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptan-4-yl]formamido}acetamide
N-(4-methyl-2-oxo-2H-chromen-7-yl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carboxamide
4-(dimethylamino)-N-ethyl-N-[2-(2-fluorophenoxy)ethyl]benzamide
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-methyl-2-phenylpropan-1-one
1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-methyl-4-(4-methylphenyl)piperazine
N-methyl-N-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}thian-4-amine
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]thieno[3,2-d]pyrimidin-4-amine
5-fluoro-N4-methyl-N2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-2,4-diamine
N-{[3-(benzyloxy)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
3-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-3,9-diazaspiro[5.6]dodecan-10-one
N-{2-[1-(3,4-difluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-4-fluorobenzamide
3-(2-chloro-4-fluorophenyl)-1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-methylurea
3-cyclopropyl-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
3-methyl-7-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
8-[(3-fluorophenyl)methyl]-3-{2-[methyl(2-methylpropyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-cyclohexylpiperidin-3-yl)-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
2-(1H-1,3-benzodiazol-2-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]acetamide
4-methoxy-3-{4-[1-(piperidin-1-yl)ethyl]phenyl}benzamide
(3S,4S)-4-cyclopropyl-1-(4-sulfamoylbenzoyl)pyrrolidine-3-carboxylic acid
3-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-indole
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
2-[5-(2-chloro-4-fluorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
1-(1H-pyrazol-1-ylmethyl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropane-1-carboxamide
3-(methoxymethyl)-N-[3-(propan-2-yloxy)propyl]benzamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-[(naphthalen-2-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-[(dimethylcarbamoyl)amino]acetamide
2-(4-fluorophenyl)-2-{[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]formamido}acetic acid
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-propylpyrrolidin-3-yl]-2-methyl-1,3-benzothiazole-5-carboxamide
6-[(diethylamino)methyl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(furan-2-ylmethyl)piperidine-4-carboxamide