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5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-1-(naphthalen-2-ylmethyl)azepan-2-one
1-(2-{4-[(4-methoxynaphthalen-1-yl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
4-({1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-2-yl}methyl)morpholine
N-(2-chloro-6-methylphenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-(3-phenylpropyl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2S,4S)-4-amino-N,N-diethyl-1-(3,3,3-trifluoropropanesulfonyl)pyrrolidine-2-carboxamide
N-[(3S,4R)-4-methoxyoxolan-3-yl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
2-(pyrrolidin-1-yl)-N-[(4-sulfamoylphenyl)methyl]pyrimidine-5-carboxamide
2,3-dimethoxy-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
3-{[2-(hydroxymethyl)azepan-1-yl]methyl}-1,2-dihydroquinolin-2-one
5-methyl-N-(2-methylpropyl)-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-1-(thiophen-2-yl)urea
(3S,4R)-4-(2-methylphenyl)-1-(6-methylpyridine-2-carbonyl)pyrrolidine-3-carboxylic acid
2-(dimethylamino)-N-({3-[(dimethylamino)methyl]phenyl}methyl)-2-(3-fluorophenyl)-N-methylacetamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}quinoline-6-carboxamide
1-[(2-chlorophenyl)methyl]-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-(2-chlorophenyl)-4-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}pyrimidine
4-(5-acetylthiophene-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
2-(dimethylamino)-2-(3-fluorophenyl)-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}acetamide
N-[2-(azepan-1-yl)-2-phenylethyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-fluoroethyl)acetamide
N-[(5-methylthiophen-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-benzyl-3-ethyl-1-(6-methylpyridazin-3-yl)-1,4-diazepan-5-one
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]acetamide
9-(3-ethyl-1H-indole-2-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
methyl (1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
4-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
4-{imidazo[1,2-a]pyridine-6-carbonyl}-2-(piperidin-1-ylmethyl)-1,4-oxazepane
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
N-(3-methoxypropyl)-1-methyl-N-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-amine
(1S,5R)-6-(2-methoxyethyl)-3-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
(benzylsulfamoyl)({[5-(pyridin-2-yl)thiophen-2-yl]methyl})amine
1-(2-methoxyacetyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carboxamide
1-{[5-(2,6-dimethylhept-5-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,3-dimethylurea
1-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
4-[5-(dimethyl-1,3-thiazole-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
4-{[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}benzoic acid
2-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]-N-ethylacetamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]propanamide
N-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]methanesulfonamide
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
5-{3-[(2-fluorophenyl)formamido]propanoyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid