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1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
N-cyclopropyl-N-(thiophen-3-ylmethyl)morpholine-2-carboxamide
2-benzyl-9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)(methyl)amino]-N-methylpropanamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-cyclohexyl-4-(5-methyl-1-benzofuran-2-carbonyl)-1,4-diazepane
N2-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-N1-(pyridin-3-yl)ethane-1,2-diamine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylthiophene-3-carboxamide
5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-(quinolin-6-ylmethyl)-1-benzofuran-2-carboxamide
[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[4-(pyridin-2-ylmethoxy)phenyl]methyl}amine
2-(3,4-dichlorophenyl)-1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
(1s,4s)-4-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)cyclohexan-1-ol
N-ethyl-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-(4-methyl-5-phenylthiophene-2-carbonyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
dimethyl[1-(5-methyl-4-phenyl-1H-imidazol-1-yl)pentan-2-yl]amine
2-{[(2E)-3-(furan-2-yl)prop-2-en-1-yl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
6-(2-chlorophenyl)-2-(3-methylpiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[2-(furan-2-yl)ethyl]-7-(oxolane-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(oxolan-2-yl)-3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
methyl 2-(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
4-[5-(2,6-difluoro-3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]butan-2-ol
4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-cyclohexylpiperazin-2-one
2-methyl-4-[(1E)-pent-1-en-1-yl]-6-(1H-pyrazol-1-yl)pyrimidine
N-methyl-N-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)methanesulfonamide
1-(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)piperidin-3-ol
2-(2-cyclopropylpyrimidin-5-yl)-N-ethyl-6-methyl-N-(propan-2-yl)quinoline-4-carboxamide
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyrrolidin-1-yl)ethan-1-one
4-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-N,N-dimethyl-4-oxobutanamide
2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-4-(pyridin-3-yl)pyrimidine
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
4-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]benzene-1-sulfonamide
2-({methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}methyl)benzonitrile
2-methoxy-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]phenol
1-{1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}pyrrolidin-2-one
5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
(3-{[1-(1-cyclobutanecarbonylpiperidin-4-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
1-cyclobutanecarbonyl-4'-methyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-2-sulfonyl)piperidine
N-({1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}methyl)quinoline-8-sulfonamide
2-(dimethyl-1,3-thiazol-5-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(4-propyl-1,4-diazepan-1-yl)pyridine-3-carboxamide
5-(4-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-2-methyl-2H-1,2,3,4-tetrazole
(1S,5R)-6-methyl-3-{2-[3-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(diethylamino)-N-(furan-2-ylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-chloro-3-{[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-pyrazole
6,7-dimethoxy-3-[(4-methyl-1H-imidazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
methyl[2-methyl-2-(morpholin-4-ylmethyl)propyl][1-(4-methylpyridin-2-yl)propan-2-yl]amine
methyl 6-[(3aS,6aR)-2-oxo-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-3-carboxylate
1-(2-fluorophenyl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}cyclopropane-1-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide