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4-({4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
1-[1'-(2,3-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
4-(3-{3-[3-(6-methoxypyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}propyl)morpholine
7-cyclohexyl-2-[4-(propan-2-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
4,4-difluoro-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidine
2-ethyl-7-methoxy-4-(quinolin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(cyclopropylmethyl)-2-oxo-3-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
2-[4-(1-methyl-1H-indole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[(4-chlorophenyl)methyl]-N-[3-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
1-[(2-methoxyphenyl)methyl]-4-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
4-methyl-2-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-[3-(2-methoxyphenyl)propyl]piperidin-4-amine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrimidin-4-amine
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
N-[2-(4-fluorophenyl)ethyl]-2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]acetamide
8-methyl-2-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-2,8-diazaspiro[4.5]decane
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-(2-{1-[(2,3-dimethyl-1H-indol-7-yl)methyl]piperidin-3-yl}ethyl)acetamide
N,8-dimethyl-3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-ethyl-5-({[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]benzonitrile
1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
2-{1-[(4-fluorophenyl)methyl]-4-[(6-fluoroquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-2-(pyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-{[1-(propan-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,3S,5S)-8-(2,6-dimethylquinoline-3-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
2-[(1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidin-4-yl)oxy]pyrimidine
1-{5-[(pyridin-3-yl)carbamoyl]furan-2-yl}-1H-imidazole-4-carboxylic acid
2-[(3,5-difluorophenyl)methyl]-8-[2-(propylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2,6-dimethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidine-4-carboxamide
7-(cyclohexylmethyl)-2-[(2-methoxypyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decane
4-ethyl-1-methyl-3-{[1-(oxolane-3-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-methylphenyl)-5-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyrimidine
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[2-(1H-pyrazol-1-yl)phenyl]methyl})amine
1-acetyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylpiperidine-4-carboxamide
3-cyclohexyl-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazole-2-carboxamide
4-({[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-2-methylbutan-2-ol
(3aS,6aS)-2-(2-methylpropyl)-5-[4-(thiophen-2-yl)butanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[4-(ethylsulfanyl)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
3-cyclohexyl-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
(1S,4S)-5-(2,2-diphenylacetyl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(2-methoxyethyl)-9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-cyclopropyl-6-(3-phenylpiperazin-1-yl)pyrimidine
2-{4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-1,4-diazepan-1-yl}-N,N-dimethylacetamide
2-(dimethyl-1,2-oxazol-4-yl)-N-(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)pyrrolidine-1-carboxamide