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2-methyl-8-(4-methylpyrimidin-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-(thiomorpholin-4-yl)butan-1-one
N-(1-phenylethyl)-3-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propanamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[(4-methoxyphenyl)methyl]amino}methyl)piperidin-2-one
2-[(3,4-difluorophenyl)methyl]-8-(3-hydroxypropanoyl)-2,8-diazaspiro[4.5]decan-3-one
1-[5-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
2-(2-{[3-(hydroxymethyl)-3-propylpiperidin-1-yl]methyl}phenoxy)acetic acid
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-hydroxy-N-(oxolan-2-ylmethyl)propanamide
N-(1-benzofuran-2-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(cyclohexylmethyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
1-cyclobutanecarbonyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]piperidine
2-{[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
1-cyclopentyl-N3-ethyl-N3-(2-methylprop-2-en-1-yl)-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-{1-[2-(propylsulfanyl)acetyl]piperidin-3-yl}benzoic acid
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(thiolan-3-yl)pyridin-2-amine
1-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(adamantan-2-yl)-4-methyl-1,4-diazepan-5-one
(3S,4R)-1-[3-(methylsulfanyl)propyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-({1-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}methyl)morpholine
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}carbamate
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}-1,3-oxazole
N-(2-hydroxyethyl)-3-propyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
2-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
2-[2-(pyridin-4-yl)ethyl]-9-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-(hydroxymethyl)-1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
7-(cyclohexylmethyl)-2-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-(2,3-dichlorophenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-1,2,3-triazole
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidin-2-amine
(3aR,7aS)-2-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
ethyl(oxan-4-ylmethyl)(quinolin-4-ylmethyl)amine
4-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-(5-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-methyl-2-(methylsulfanyl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
1-[1-(furan-3-carbonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
N-(4-methoxy-2-methylphenyl)-3-[1-(pyridine-4-carbonyl)piperidin-3-yl]propanamide
1-methyl-4-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,4-dihydroquinoline-3-carboxamide
methyl 3-[(3S,4R)-1-[(3-hydroxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
2-methyl-N-{2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]phenyl}propanamide
(3R,4S)-N-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1-methanesulfonyl-4-propylpyrrolidin-3-amine
(3S,4S)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(2R,3R,6R)-3-(4-methoxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-methyl-1H-pyrazole-4-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
3-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one