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1-tert-butyl-N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-[(3S,4R)-1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-(3,5-dimethyl-4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
2-[1-(3-fluorophenyl)-5-[(2-oxo-1,2-dihydropyridin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
methyl 1-(2-methoxyethoxy)-2-oxo-8-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
N-cyclopropyl-4-{[(4-methylphenyl)amino]methyl}-N-propylbenzamide
2-methanesulfonamido-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
cyclohexyl[4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
4-[7-(3-cyclopentylpropanoyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)ethan-1-ol
1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}isoquinoline
N-[2-(dimethylamino)ethyl]-5-(oxolane-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3aR,6aR)-2-cyclopentyl-N-[2-(4-hydroxyphenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-{[(6-ethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-ol
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(furan-2-ylmethyl)-6-oxo-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(3-methoxyphenyl)-4-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]piperazin-2-one
2-(4-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}morpholin-3-yl)acetic acid
4-[(2-chloro-6-fluorophenyl)methyl]-3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]piperazin-2-one
(3S,4S)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(naphthalen-2-yl)piperidin-3-ol
1-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
5-[1-(methoxymethyl)cyclobutyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
3-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
3-[(5-fluoroquinazolin-4-yl)amino]-1-methylpyrrolidin-2-one
2-{[(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
N-cyclopropyl-4-methyl-2-(4-methylpiperazin-1-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}pyrimidine-5-carboxamide
N-(3,5-dimethoxyphenyl)-3-[1-(thian-4-yl)piperidin-3-yl]propanamide
4-{1-[4-(morpholin-4-yl)butanoyl]piperidin-3-yl}benzoic acid
1-ethyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxamide
1-[2-(3-methoxyphenyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-(4-{5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-6-methylpyridine
(1S,5R)-3-(3-methanesulfonylpropanoyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl[(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl](1,2-oxazol-3-ylmethyl)amine
1-[(5-ethylfuran-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2,4-difluoro-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzene-1-sulfonamide
3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
(but-2-yn-1-yl)[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](furan-2-ylmethyl)amine
2-[(4aS,7aR)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
methyl 6-({[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
5-ethyl-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,2,4-oxadiazol-3-amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide