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1,3-dimethyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
[(dimethyl-1,2-oxazol-4-yl)methyl][(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
4-methyl-5-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}thiophene-2-carboxamide
3-methyl-8-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl 4-{[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-3-(pyrimidin-2-yloxy)benzamide
N-[(2R,3R)-1'-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-6-azaspiro[2.5]octane-1-carboxamide
4-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methylacetamido]butanoic acid
(3aR,5S,6S,7aS)-2-{[2-(trifluoromethoxy)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-(1-cycloheptylpiperidin-3-yl)-3-(pyridin-4-yl)propanamide
5-chloro-N,4,6-trimethyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-ol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pent-4-enamide
5-methoxy-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-methyl-1H-indole
1-(4-{[2-(1H-imidazol-4-yl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
2-chloro-N-{1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
3-[(3R,4S)-1-(4-chlorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[(1-hydroxycyclohexyl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-6-methylquinoline
4-({4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenol
[3-(dimethylamino)-2,2-dimethylpropyl][(5-ethylpyridin-2-yl)methyl]methylamine
2-methoxy-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
5-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
1-cyclopentyl-3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[(2-methoxyphenyl)methyl]urea
N-(propan-2-yl)-2-(pyridin-3-yl)pyridine-4-carboxamide
1-[(4-hydroxy-3-methylphenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amine
2-ethoxy-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyridine
3-{[1-(1-benzylpiperidin-4-yl)piperidin-3-yl]formamido}propanamide
5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}-1H-1,2,3,4-tetrazole
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
1-{[3-(3-phenylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-(4-methylphenoxymethyl)-1-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-1H-1,3-benzodiazole
2,3-dimethyl-N-[(4-sulfamoylphenyl)methyl]quinoxaline-6-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(4aR,7aS)-1-ethyl-4-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-methylbenzamide
8-[(4-acetylphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(dimethyl-1,2-oxazole-4-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
6-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
1-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-2-phenylethane-1,2-dione
N,5-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}propanamide
4-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-1λ6-thiane-1,1-dione