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N-[3-(azepan-1-yl)-2-hydroxypropyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
2-(2,2-dimethylpropanamido)-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-5-methylthiophene-3-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]methyl}-1-ethenyl-1H-pyrazole-4-carboxamide
3-(1H-imidazol-1-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)propanamide
N-{3-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]phenyl}acetamide
1-(2-chlorophenyl)-4-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)piperazin-2-one
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-methylbenzoyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3R,4S)-1-[4-(1H-imidazol-1-yl)benzoyl]-4-(3-methoxyphenyl)pyrrolidin-3-amine
2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
1-(4-fluorophenyl)-6,6-dimethyl-N-[(6-methylpyridin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[2-({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)ethyl]-3,4-dihydroquinazolin-4-one
N-(3-fluorophenyl)-4-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}benzamide
3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-{2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{2-[cyclopentyl(methyl)amino]ethyl}-4-hydroxy-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
5-[(1-benzothiophen-2-ylmethyl)amino]-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 4-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)carbamoyl]amino}benzoate
N-methyl-2-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)acetamide
1-[3-(4-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl}pyridin-2-yl)phenyl]ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-(1-{[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
methyl[(2-methyl-1,3-oxazol-4-yl)methyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
3-methyl-5-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-({5-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
6-cyclopropyl-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
3-[2-(dimethylamino)ethyl]-8-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3-benzyl-1H-pyrazol-5-yl)-1-(oxane-4-carbonyl)piperidine
(3S,4S)-1-(1-phenylcyclopropanecarbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
6,7-dimethoxy-2-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazine-2-carboxylic acid
8-[(4-methanesulfonylphenyl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-{1-[5-(3-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}pyrrolidin-2-one
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)-N-methylacetamide
N-[4-(4-{[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
methyl 4-methoxy-3-[({1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}carbamoyl)amino]benzoate
5-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}-2-methylpyrimidin-4-ol
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[4-(4-phenylazepane-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-chlorophenyl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
4-(3-phenyl-1H-1,2,4-triazol-5-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dimethoxybenzamide
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-8-propanoyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(5S,9aS,9bS)-5-(3-hydroxy-4-methoxyphenyl)-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(butan-2-yl)[(4-methyl-1H-imidazol-5-yl)methyl](thiophen-3-ylmethyl)amine
6-{4-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-9H-purine
1-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one