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N-(2H-1,3-benzodioxol-5-ylmethyl)-N,1,5-trimethyl-1H-pyrazole-3-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,2-dimethylmorpholine
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(pyridin-4-yl)-decahydroisoquinoline
2-({[4-(methylsulfanyl)phenyl]methyl}({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amino)ethan-1-ol
ethyl 1-(1-ethylpiperidin-4-yl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({[4-(methylsulfanyl)phenyl]methyl}(pyridin-4-ylmethyl)amino)ethan-1-ol
methyl 5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-(carbamoylmethyl)-N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(2R,6S)-2,6-dimethyl-4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)morpholine
1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-(pyrimidin-2-yl)-1,4-diazepane
N-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
1-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-chloro-N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-1-methyl-1H-pyrazole-5-carboxamide
4-{3-cyclopropyl-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
6-(4-ethoxypiperidine-1-carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(trifluoromethyl)cyclopropane-1-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
4-(2-methoxyphenyl)-2-methyl-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperazine
5-({2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}methyl)-N,N-dimethylfuran-2-carboxamide
2-(3,4-dimethoxyphenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
N-methyl-5-({4-[5-(oxan-2-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}methyl)furan-2-carboxamide
(5S,9aS,9bS)-5-[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-fluoro-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-2-amine
5-{[methyl({[3-(2-{4-[4-(trifluoromethoxy)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(pyridin-3-ylmethyl)piperazine
N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
methyl 3-{methyl[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}benzoate
N-[(2,5-dimethylphenyl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
4-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]oxane-4-carbonitrile
(3S,4R)-1-(2-cyclopentylacetyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-({4-[3-(benzyloxy)azetidin-1-yl]-6-methylpyrimidin-2-yl}amino)phenol
(1R,5R)-3-benzoyl-6-(thiophen-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-benzyl-8-[(4-hydroxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(2-phenylpyrimidin-5-yl)methyl]-decahydro-2,7-naphthyridine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
[(3R,4R)-1-[(6-methylpyridin-2-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3S)-3-(3-methoxyphenyl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine
1-[cyclohexyl(methyl)amino]-3-[3-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
4-methyl-6-(pyridin-4-yl)-2-(pyrrolidin-1-yl)pyrimidine
4-(3-methyl-1,2,4-oxadiazol-5-yl)-N-(pyridin-4-ylmethyl)aniline
3-{[8-(1,3-benzothiazol-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyridin-2-amine
6-[3-(hydroxymethyl)piperidin-1-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
methyl 3-chloro-4-{[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]amino}benzoate
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}ethan-1-one
2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(piperidin-4-yl)-N-propylpyrimidin-4-amine