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3-(3-chlorophenyl)-N-(3-methyl-1-propyl-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
8-chloro-2-[(4-hydroxyazepan-1-yl)methyl]quinolin-4-ol
1-[(2,4-difluorophenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-(3-chloro-2-methylphenyl)-N'-methyl-N'-(oxan-4-yl)butanediamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
[(3R,4R)-1-(2,6-difluoro-4-methoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(2-phenylbenzoyl)pyrrolidin-3-yl]methanol
{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}({2-[2-(trifluoromethyl)phenyl]ethyl})amine
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-ethylbutanamide
1-ethyl-4-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N2,N2-dimethylpyrazine-2,3-diamine
3-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]-1-[1-(2-methylphenoxy)propan-2-yl]urea
6-(3-fluorophenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
2-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)methyl]quinolin-4-ol
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
(4S)-1-(5-ethylthiophene-2-carbonyl)-3,3,4-trimethylpiperidin-4-ol
2-methyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1-benzofuran-5-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
5-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-methyl-N-[(3R)-pyrrolidin-3-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
3-(5-ethyl-1,2-oxazole-3-carbonyl)-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}acetamide
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(pyridin-4-ylmethyl)amine
1-{3-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propyl}-1H-pyrazole
1-(2-{2-[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-4-methyl-1H-1,2,3-triazole
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-[3-(4H-1,2,4-triazol-4-yl)phenyl]thiophene-2-carboxylic acid
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
2-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]benzonitrile
2,8-dimethyl-3-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}quinoline
3-amino-N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-1,2,4-triazole-5-carboxamide
2-(2-methoxyethyl)-8-[(1-methyl-1H-indol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
N-ethyl-5-[1-(piperidin-1-yl)ethyl]-N-(pyridin-4-ylmethyl)furan-2-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[2-(2-methoxyphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
8-fluoro-2-{[(1r,5r)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]methyl}quinolin-4-ol
2-(dimethylamino)-8-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
7-(1,3-benzothiazol-2-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-({1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
4-{1-[1-(pyrazin-2-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}quinoline
[5-(1-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-imidazol-2-yl)furan-2-yl]methanol
3-(3,4-dimethoxyphenyl)-N-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
3-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1,2-benzothiazole
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]piperidine