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2-[(4-fluorophenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]morpholine
2-(azocan-1-yl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(3S,5S)-1-[(2,4-difluorophenyl)methyl]-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
2-{3-[1-(2-fluoroethyl)-1H-pyrazol-3-yl]phenyl}-4,6-dimethoxypyrimidine
5-(9H-fluoren-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-(quinoline-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(2-chloro-4-fluorophenoxymethyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-methyl-3-(naphthalen-2-ylmethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-benzoyl-6-(3-propyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]methyl}benzonitrile
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyrrolidin-1-yl)benzamide
N-[(2R,3R)-2-ethoxy-1'-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
[(3R,4R)-1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-{6-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridin-3-yl}ethan-1-one
2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-4-(2-methoxyphenyl)pyrimidine
2-({[(3R,4R)-1-(2-chloro-5-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
7-methoxy-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(dimethylamino)ethyl]-3-[5-(pyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
3-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
N-methyl-5-{1-[2-(6-methyl-1-benzofuran-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N3-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-methyl-5-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-5-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(6-ethylpyrimidin-4-yl)piperidine-4-carboxylic acid
4-[(1-phenylbutyl)carbamoyl]pyridin-1-ium-1-olate
(3R,4R)-4-ethyl-1-(6-methoxypyrimidin-4-yl)piperidine-3,4-diol
6-ethyl-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
5-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(2-methylpropanoyl)-2,7-diazaspiro[4.5]decan-6-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(3-methylthiophen-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{2-[5-(8-methoxyquinolin-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-(2-chloro-6-fluorophenyl)-1-{imidazo[1,2-a]pyridin-3-ylmethyl}-1H-imidazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(5-oxopyrrolidine-3-carbonyl)piperazin-2-one
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)propanamide
N-[(3R,4S)-1-cyclopentanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-2-phenoxyacetamide
2-({[2-(benzylamino)pyrimidin-5-yl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-phenylmethanesulfonylpiperidine
4-[2-(dimethylamino)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
3-(5-{3-[1-(dimethylamino)ethyl]phenyl}-4-phenyl-1H-imidazol-1-yl)propanamide
1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-8-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-propylpiperidine
N-[2-(methylsulfanyl)ethyl]-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(2S)-2-({1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-4-methylpentanamide
N-[2-(2-ethoxyphenoxy)ethyl]-2-methanesulfonyl-N-methylacetamide
3-methyl-6-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}pyridazine
3-benzyl-4-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperazin-2-one