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1-(2-{[4-(ethylamino)pyrimidin-2-yl](methyl)amino}ethyl)piperidin-2-one
(1R)-3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-phenylpropan-1-ol
1-{4-[(cyclohexylamino)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
{[(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-amino-6-{4-[(5-propylfuran-2-yl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
6-methyl-2-(4-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
[(3-methoxyphenyl)methyl][3-(methylsulfanyl)butyl](prop-2-en-1-yl)amine
2-({[2-(2-ethoxyphenoxy)ethyl](methyl)amino}methyl)-6-methylpyridin-3-ol
1-[1-(5-fluoro-2-methoxybenzoyl)piperidin-4-yl]piperidin-3-ol
5-methoxy-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)furan-2-carboxamide
4-(5-{1-[(2-methoxyphenyl)methyl]-1H-imidazol-2-yl}pyrimidin-2-yl)morpholine
methyl[(3-methylthiophen-2-yl)methyl]{[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
2-amino-4-[(furan-2-ylmethyl)(methyl)amino]quinazoline-6-carboxylic acid
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]propan-1-one
5-methoxy-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(1H-pyrazol-3-yl)pyridine
1-{2-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-4-methylpiperazine
(1S,5R)-3-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(5-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-yl}-1,2,4-oxadiazol-3-yl)pyridine
2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
8-chloro-2-(4-cyclohexylpiperazine-1-carbonyl)quinoline
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(4aS,8aR)-6-({3-[(dimethylamino)methyl]phenyl}methyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-6-ethyl-N,2-dimethylquinoline-4-carboxamide
1-[(3-{[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-2-yl)piperazine
methyl (1R,3S,3aR,6aS)-1-ethyl-3-(6-methylpyridin-2-yl)-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(3aR,7aS)-2-[(1-benzyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
[3-(4-cyclopentylpyrimidin-2-yl)phenyl]methanamine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(2-methyl-6-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1-propylurea
5-ethyl-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]pyrimidin-2-amine
3-(1-methylcyclopropyl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
(1R)-1-[1-(3-chloro-2-methylphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
2-{2-[5-(5-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrazine
4-methyl-2-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}phenol
4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(phenylsulfanyl)propyl]pyrimidin-2-amine
N-[4-(4-methoxypiperidine-1-carbonyl)phenyl]ethane-1-sulfonamide
2-(adamantan-1-yl)-4-hydroxy-N-[(5-methylpyrazin-2-yl)methyl]pyrimidine-5-carboxamide
6-methoxy-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(furan-2-yl)ethane-1,2-dione
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1R,9S)-5-amino-3-(3-fluoro-5-methylphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-{1-[(3,4-difluorophenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-yl}ethan-1-ol
N-[4-(2-ethyl-1-benzofuran-3-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]acetamide