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2-{3-[(1-methylpiperidin-4-yl)methyl]-5-[(1S)-1-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
(4aS,8aR)-1-(4-hydroxybutyl)-6-[3-(pyridin-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N1,N1-dimethyl-N4-[1-(2-phenylethyl)piperidin-3-yl]piperidine-1,4-dicarboxamide
4-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
dimethyl(2-{2-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-3-amine
N'-{[(1R,2R)-2-hydroxycyclohexyl]methyl}-N-[2-(methylsulfanyl)phenyl]butanediamide
3-cyclopropyl-5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-1-(3-fluorophenyl)-1H-1,2,4-triazole
N-(2-phenoxyethyl)-2-propanoyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methyl-2-phenylpyrimidine
1-[(4-methylphenyl)methyl]-5-(1H-pyrrol-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
7-methanesulfonyl-N,4-dimethyl-N-[2-(pyrrolidin-1-yl)ethyl]quinazolin-2-amine
N4-ethyl-N2-methyl-N2-[(4-methyl-1H-imidazol-2-yl)methyl]pyrimidine-2,4-diamine
N-[(1S,2R)-1-carbamoyl-2-hydroxypropyl]-N'-(2,4-dimethylphenyl)propanediamide
N-ethyl-6-methyl-N-(2,2,2-trifluoroethyl)imidazo[1,2-a]pyridine-2-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-3-amine
6-methyl-4-(2-oxo-2-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}ethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-(6-chloro-2-methylpyridin-3-yl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
3-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propanamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1H-imidazol-1-yl)ethyl]-N-methylbenzamide
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-[5-({7-methyl-12-oxo-3,7,11-triazaspiro[5.6]dodecan-3-yl}methyl)furan-2-yl]benzonitrile
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-(2-ethoxyethyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(4-chlorophenyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
3-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-N-(propan-2-yl)propanamide
5-(2-chloro-4-fluorophenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1,2-oxazole-3-carboxamide
3-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-2-(4-hydroxyphenyl)acetic acid
2-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
5-(3,4-dimethoxyphenyl)-1-(oxan-2-ylmethyl)-4-phenyl-1H-imidazole
3-[(3-chlorophenyl)methyl]-N-[1-(thiophen-2-yl)propan-2-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-4-(morpholin-4-yl)-N-(pyridin-3-ylmethyl)benzamide
1-(furan-2-ylmethyl)-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]piperidine-4-carboxamide
(1S)-1-[1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethan-1-ol
2-(2-{[cyclopropyl(1-methylpiperidin-4-yl)amino]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
5-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
(1S,5R)-3-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methoxyquinoline-4-carboxamide
4-[(7-hydroxyquinolin-3-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-1,4-diazepan-5-one
(1R,2S,6R,7S)-4-(1H-pyrazole-3-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
[1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
6-ethoxy-3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
6-[({[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
(3R,5S)-1-benzyl-N-(2,3-dihydro-1H-inden-5-yl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
(1R,3S)-7-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-7-azaspiro[3.5]nonane-1,3-diol
1-[(3-acetylphenyl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-(3-fluorophenoxy)-1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one