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2-[1-(3,5-dichloro-4-methylbenzoyl)piperidin-2-yl]pyridine
9-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1H-indol-2-yl)phenyl]-1-(thian-4-yl)piperidine-4-carboxamide
(3aS,6aS)-2-(2-methoxyacetyl)-5-[(2-methylnaphthalen-1-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[3-(furan-2-yl)-3-phenylpropyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
8-{[3-(furan-2-yl)phenyl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-methanesulfonyl-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}furan-2-yl)methyl]-1H-imidazole
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-4-(pyridin-3-yl)pyrimidin-2-amine
(4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
[3-(cyclopropylmethyl)-1-(5,6-dimethylpyrazin-2-yl)piperidin-3-yl]methanol
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenol
3-ethyl-8-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-({4-[2-methoxy-5-(propan-2-yl)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-4-methyl-1H-imidazole
4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
N,1-dimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1H-1,3-benzodiazole-5-carboxamide
2-ethyl-6-methyl-5-{[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydropyrimidin-4-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1-methyl-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 3-cyclohexaneamido-5-({imidazo[2,1-b][1,3]thiazol-6-ylformamido}methyl)benzoate
(4aS,8aR)-1-(3-hydroxypropyl)-6-(5-methylthiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
4-(3,6-dimethylpyrazin-2-yl)-2-(morpholin-4-ylmethyl)phenol
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[2-(pyridin-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(3S,9aR)-8-(3-chlorobenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-(dimethylamino)-4-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}pyrimidine-5-carboxamide
2-{4-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]morpholin-3-yl}acetic acid
propan-2-yl 4-[2-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)ethyl]piperidine-1-carboxylate
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazol-1-yl}acetic acid
propan-2-yl 4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carboxylate
3,5-dimethyl-4-oxo-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-5-(3-fluorophenyl)-1,2,4-triazin-3-amine
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-[(2-fluoro-5-methylphenyl)methyl]-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
1'-(3-ethyl-1,2-oxazole-5-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1,9-dimethyl-4-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-1,4,9-triazaspiro[5.5]undecane
1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butane-1,2-dione
4-[5-(3,4-dimethylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
1-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-4-(1H-imidazol-1-yl)butan-1-one
4-[1-(propan-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)morpholine-2-carboxamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
5-fluoro-2-[1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
(4aS,8aR)-6-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-(cyclohex-3-en-1-ylmethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide