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1-cyclobutanecarbonyl-4-(2-methyl-1-benzofuran-7-carbonyl)-1,4-diazepane
(3R,4R)-1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
3-[1-(8-fluoroquinoline-2-carbonyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-[2-(pyridin-2-yl)ethyl]pyridin-2-amine
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(2-methylphenyl)methyl]carbamoyl}pyrrolidine-2-carboxylate
1'-[1-(propan-2-yl)piperidine-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(4-methoxy-2-methylphenyl)-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-3-yl}propanamide
(3E)-N-[1-(6-methoxynaphthalen-2-yl)ethyl]pent-3-enamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
4-(3-cyanopyridin-2-yl)benzamide
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-(furan-3-yl)-4-phenyl-1H-imidazole
5-{[4-(3-ethylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}-2-methyl-1,3-benzothiazole
5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
6-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]quinoxaline
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-[4-(2,3-dichlorophenyl)-8-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methoxyacetamide
2-(6-methoxypyridin-3-yl)-2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]acetic acid
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-({6-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridin-3-yl}methyl)acetamide
8-(2-hydroxy-3-methoxybenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2,6-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-3-carboxamide
3-[methyl({2-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyrimidin-4-yl})amino]propane-1,2-diol
(1S,5R)-6-benzyl-3-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)oxolane-2-carboxamide
1-(propan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3S)-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
N,5-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-cyclopropyl-9-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2,6-dimethylpyrimidine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-(pyrazin-2-yl)propan-1-one
(1S,5R)-6-(5-methylthiophene-2-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3-methylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-(4-hydroxyphenyl)propan-1-one
N,N-dimethyl-3-[2-(methylsulfanyl)benzoyl]piperidine-1-sulfonamide
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-propyl-1H-pyrazole-5-carboxamide
3-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1-(4-methoxyphenyl)urea
2-(2,5-dioxoimidazolidin-4-yl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}acetamide
N-(2-propoxypropyl)-3-(1H-pyrazol-4-yl)benzamide
1-{2-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2-methyl-1H-1,3-benzodiazole
2-(4-{[2-(methoxymethyl)piperidin-1-yl]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-[(2-methoxyphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1-propyl-1H-1,2,4-triazole
2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane
N-[(3R,4R)-3-hydroxy-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl]pyridine-3-carboxamide
(3R,4S)-1-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}-4-phenylpyrrolidin-3-amine
3-[(4-methanesulfonylphenyl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran