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N-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylpyrrolidin-3-amine
5-cyclopropyl-N,N-diethyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-(methylamino)pyridine-4-carboxamide
methyl 3-(3-cyclohexylpropanoyl)-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-6-[2-(pyrrolidin-1-yl)ethyl]pyridine-3-carboxamide
6-[4-(methoxymethyl)piperidin-1-yl]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
(1R,5S,6S)-6-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
1-methyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-(morpholin-4-yl)-1H-1,3-benzodiazole
4-(azepane-1-carbonyl)-7-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
4-fluorophenyl (7R,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-{[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]sulfamoyl}-N,N-dimethylbenzamide
1-cyclohexyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidine-4-carboxamide
N-({1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]pyrrolidin-3-yl}methyl)azetidine-3-carboxamide
6-methoxy-N,3-dimethyl-N-(quinolin-6-ylmethyl)-1-benzofuran-2-carboxamide
7-[(4,4-difluoropiperidin-1-yl)methyl]-2,3-dimethyl-1H-indole
ethyl 2-(1-{5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazol-4-yl}-N-methylformamido)acetate
1-[(4-ethoxyphenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(2R,3R,6R)-5-(2-methoxyethyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(N-methylmethanesulfonamido)ethyl]-5-(4-methylphenyl)furan-2-carboxamide
3-({1-[2-(benzyloxy)acetyl]pyrrolidin-3-yl}methyl)benzamide
3-[1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)-N-methylformamido]propanamide
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(2,2,2-trifluoroethyl)piperazine
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
6-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methoxy}quinoline
(1R,5S,8S)-8-methoxy-3-[(3-methyl-1-benzofuran-2-yl)methyl]-3-azabicyclo[3.2.1]octane
(2R)-2-[(5-methylhexan-2-yl)amino]-3-phenylpropan-1-ol
1-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-(4-methylbenzenesulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-[(4aR,8aS)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-decahydro-1,6-naphthyridin-6-yl]-3-(pyridin-3-yl)propan-1-one
N-methyl-6-(4-methylquinolin-2-yl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-[4-(hydroxymethyl)phenyl]-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-cyclohexyl-6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-N-methylpyridin-2-amine
3-[2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
9-(2-ethoxypropanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-(pyridin-2-ylmethyl)piperidin-4-amine
5-(1-benzofuran-5-yl)-3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-ethyl-N-(2-methylprop-2-en-1-yl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
1-methyl-9-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}morpholine-2-carboxamide
{5-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
N-[2-(dimethylamino)ethyl]-2-methyl-N-{[8-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide
5-(4-methyl-1H-pyrazol-1-yl)-N-(pyridin-3-yl)furan-2-carboxamide
2-({[3-(2-methoxyethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-thiadiazole
1-[(4-fluorophenyl)methyl]-3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
1-ethoxy-3-[5-(2-fluoro-3-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propan-2-ol
9-(2-hydroxyethyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one