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1-methyl-3-[4-(2-methylphenyl)-3-oxopiperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[4-(piperidine-1-sulfonyl)-1,4-diazepan-1-yl]ethan-1-one
3-[3-(oxolan-3-yl)-5-(1H-pyrrol-3-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-[1-(1-butanoylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
4-[(3,4-dimethoxypyridin-2-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
2-[(cyclopropylmethyl)sulfanyl]-1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-methyl-4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-(3-methanesulfonamidophenyl)-3-(oxolan-2-ylmethyl)-3-propylurea
1'-(2,6-dimethylpyrimidine-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(2-phenylpropyl)piperidine
10-methoxy-5-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-(4-{[(1S)-1-phenylpropyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-[3-(methylsulfanyl)phenyl]-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
1-(2-aminoethyl)-N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-[5-(methoxymethyl)thiophene-2-carbonyl]-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
1-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-5-one
N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]thiophene-2-carboxamide
5-(methoxymethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}thiophene-2-carboxamide
1'-(5-phenyl-1,2-oxazole-3-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
4-hydroxy-1-(2-methylquinolin-4-yl)piperidine-4-carboxylic acid
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
N-methyl-2-[4-(7-methyl-1H-indol-3-yl)-1H-pyrazol-1-yl]acetamide
5-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}thiophene-2-sulfonamide
2-(phenylamino)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
(4aS,7aR)-1-[2-(methylsulfanyl)acetyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-1-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]-2-methylpropan-1-one
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-methoxy-1-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydropyridin-2-one
3-{1-[(4-methanesulfonylphenyl)methyl]piperidin-3-yl}benzoic acid
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
N-(2,3-dihydro-1H-inden-2-yl)-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2,4-dimethoxy-6-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
2-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-6-fluoroquinolin-4-ol
N-[2-(dimethylamino)ethyl]-N-{[7-fluoro-2-(2-methylphenyl)quinolin-3-yl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
4-[6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]morpholine
N-{3-[(dimethylsulfamoyl)amino]phenyl}-3-(propoxymethyl)pyrrolidine-1-carboxamide
N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)-2-(pyrrolidin-3-yl)acetamide
2,3-dimethyl-5-{1-oxa-7-azaspiro[3.5]nonane-7-carbonyl}benzene-1-sulfonamide
2,8-dimethyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}quinoline-4-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
1-[(2-fluorophenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)piperidine-3-carboxamide
1-butyl-4-[2-oxo-2-(5-oxo-1,4-diazepan-1-yl)-1-phenylethyl]piperazine-2,3-dione
N-[1-(1H-indol-5-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
2-({[(3R,4R)-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide