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4-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyrimidin-2-amine
3-{[1-(2-methoxybenzenesulfonyl)pyrrolidin-3-yl]methyl}benzamide
(3aS,6aS)-2-[(3-chloropyridin-4-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-6-oxo-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1,6-dihydropyridine-3-carboxamide
4-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,2,6,6-tetramethylpiperidine
2-(3-ethoxyphenyl)-5-(1H-imidazol-1-ylmethyl)pyridine
(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-2-yl)methanol
2-[9-(5-methylpyridine-3-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-(1H-imidazol-1-yl)acetamide
(1R,5R)-6-(pyridin-2-ylmethyl)-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
3-{1-[(5-cyclohexylthiophen-2-yl)methyl]piperidin-3-yl}-N-cyclopropylpropanamide
3-{[1-methyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carbonitrile
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-propyl-1H-pyrazole-5-sulfonamide
4-{[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(2S,4R)-4-amino-1-{[1-(4-methoxyphenyl)-1H-pyrrol-2-yl]methyl}-N-methylpyrrolidine-2-carboxamide
1-ethyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-5-oxopyrrolidine-3-carboxamide
1-(furan-2-ylmethyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
4-{1-[3-(pyridin-3-yl)propyl]piperidin-3-yl}benzoic acid
N-[(1-ethylpyrrolidin-3-yl)methyl]-5-(4-fluorophenyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-[2-(2-fluorophenyl)ethyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
6-methoxy-4-oxo-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}-1,4-dihydroquinoline-3-carboxamide
2-[1-(7-fluoro-2-methylquinoline-4-carbonyl)piperidin-2-yl]acetamide
3-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propanamide
3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-N-[(2-fluorophenyl)methyl]piperidine-1-carboxamide
(1s,4s)-4-{[(oxolan-2-ylmethyl)(propyl)amino]methyl}cyclohexan-1-amine
4-{1-[2-oxo-2-(piperidin-1-yl)ethyl]piperidin-3-yl}benzoic acid
ethyl 1-[2-(2-oxopyrrolidin-1-yl)acetyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-[9-(4-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(1R,3R)-3-aminocyclopentyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
N-cyclopropyl-2-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}pyridine-4-carboxamide
2-[(4-ethylcyclohexyl)formamido]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
4,5-dimethyl-6-[4-(piperidin-1-ylmethyl)piperidin-1-yl]pyrimidine
1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
(3R,4R)-4-cyclopropyl-3-methyl-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-ol
2-(3-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)ethan-1-ol
N-[2-(diethylamino)ethyl]-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-[(3-methoxyphenyl)amino]butanamide
N-(4-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}phenyl)acetamide
N-[2-(diethylamino)ethyl]-5-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-[methyl(2-phenylethyl)amino]-N-(propan-2-yl)-2,3-dihydro-1H-indene-2-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(5-methoxyfuran-2-carbonyl)pyrrolidin-3-yl]methanol