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1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
[(3R,4R)-1-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]morpholine-2-carboxylic acid
8-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1-oxa-8-azaspiro[4.5]decane
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]ethan-1-one
(2E)-N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-fluoro-6-methoxybenzamide
8-[(3,4-dichlorophenyl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-4-phenyl-1H-pyrazol-5-amine
4-methyl-5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]pyrimidin-2-amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(1H-pyrazol-1-yl)acetyl]piperidine-2-carboxamide
methyl 4-{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}piperazine-1-carboxylate
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-[2-(4-methoxyphenyl)ethyl]azepan-4-amine
7-(3-chlorophenyl)-4-{spiro[2.3]hexane-1-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(azepane-1-carbonyl)-N-[(2,3-dimethoxyphenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
8-methoxy-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(propan-2-yl)amine
5-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)ethan-1-one
5-cyclobutyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,3,4-oxadiazol-2-amine
2-(3-cyclopentyl-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
5-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-{spiro[2.4]heptane-1-carbonyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(3-ethoxypropyl)-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
ethyl 1-(2-methylpropyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(3R,5S)-5-(morpholine-4-carbonyl)piperidine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
S-(2-cyclopropanecarbonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-hydroxybutane-1-sulfonamido
propan-2-yl 3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carboxylate
2-ethyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(4-ethynylphenyl)methyl]piperidin-4-yl}oxy)benzamide
4-{[2-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]methyl}benzene-1,3-diol
3-bromo-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
(1R,5R)-6-(cyclobutylmethyl)-3-(3-ethyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{[1-(2-methylpropyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-{[7-(cyclopent-1-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-fluorobenzamide
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl}amine
3-propyl-5-[4-(1H-pyrazol-3-yl)phenyl]-1,2,4-oxadiazole
1-{2-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(furan-2-yl)-2-hydroxyethyl]acetamide
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
8-(2-methoxyacetyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[5-(4-fluorophenyl)-1,3,4-thiadiazol-2-yl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-N-ethylcyclopropanamine
3-fluoro-5-[2-methyl-4-(3-methylphenyl)-5-oxopiperazine-1-carbonyl]benzonitrile
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-{4-[4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide