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ethyl 2-[1-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)piperidin-2-yl]acetate
2-(1,2-benzoxazol-3-yl)-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}acetamide
(3S,5S)-1-(3-hydroxypyridine-2-carbonyl)-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
1-[(3aR,6aR)-3a-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methoxyethan-1-one
methyl (2S,4R)-4-(2-cyclopropylquinoline-4-amido)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-3-[(methylsulfanyl)methyl]piperidine
2-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-cyclopentyl-3-[(oxan-4-ylmethyl)sulfamoyl]benzamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
(3R,4S)-4-cyclopropyl-1-[(2,3-difluoro-4-methoxyphenyl)methyl]pyrrolidin-3-amine
(3R)-1-{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}pyrrolidin-3-ol
4-[3-(1H-imidazol-2-yl)benzoyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2,5-dioxo-6-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(pyridin-3-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
2-{[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
(3S,4R)-1-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-[2-({[2-(4-fluorophenoxy)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
4-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
7-(cyclohexylmethyl)-6-oxo-N-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
N-{2-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
3-(5-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
1-[(3-{[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(furan-2-carbonyl)piperazine
1-[2-(dimethylamino)ethyl]-3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-methyl-2-(2-phenylethyl)-1,4-dihydropyridin-4-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(3aR,6aS)-5-[(8-methoxy-2H-chromen-3-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-methylpropyl)-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
N-({1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(1-cyclopentylpiperidin-4-yl)methyl][(2,5-difluorophenyl)methyl](oxolan-2-ylmethyl)amine
4-(6-methoxypyrimidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-N-[1-(4-propylphenyl)ethyl]acetamide
(2S)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine-2-carboxamide
N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}-2,6-dimethylquinoline-3-carboxamide
2,2-dimethyl-4-[7-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholine
5-(butane-1-sulfonyl)-2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(cyclohexylmethyl)-N3-(2-hydroxy-2-phenylethyl)-N3-methyl-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(4-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}phenyl)acetamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(quinoline-7-carbonyl)piperidin-3-yl]propanoic acid
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-methanesulfonyl-1'-[(4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[1-(4-aminobutanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[(4-methylphenyl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)urea
2-(2-{[cycloheptyl(methyl)amino]methyl}phenyl)-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)imidazo[1,2-a]pyrimidine-2-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-[(4-hydroxy-2-methoxyphenyl)methyl]piperazin-2-one
N-phenyl-5-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrimidin-2-amine