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7-methyl-N-[(5-oxo-1-phenylpyrrolidin-3-yl)methyl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
methyl 5-[(2-methylbutyl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2R,4S)-4-hydroxy-1-[3-(pyridin-3-yl)propanoyl]piperidine-2-carboxylic acid
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-{3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenoxy}acetamide
2-methyl-4-phenyl-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane
N-{[4-(5-fluoro-2-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}-N-methylmethanesulfonamide
4-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}benzoic acid
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
(2S,4S)-1-benzyl-4-[(1-ethylpiperidin-4-yl)amino]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-ethylacetamide
2-amino-8-{3-[(2-methylphenyl)methoxy]phenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-1-yl)phenol
8-(1H-indol-7-ylmethyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-cyclohexyl-5-[1-(2-methoxyethyl)pyrrolidin-3-yl]-1H-1,2,4-triazole
3-methyl-1-[2-oxo-2-(2-phenylazetidin-1-yl)ethyl]-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridine-3-carboxamide
N6-benzyl-N5-methyl-N5-[4-(morpholin-4-yl)butyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(3R,9aR)-8-benzyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-4-yl)ethyl}morpholine
2-{4-[(morpholine-4-carbonyl)amino]phenyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetic acid
1-({1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(ethylsulfanyl)propanamide
(1R,5R)-6-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{[(3S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-3-hydroxypiperidin-4-yl]methyl}-3,3-diethylurea
{1-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
1-(3-cyano-4-ethoxyphenyl)-3-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]urea
4-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4H-1,2,4-triazole
3-{1-[3-(hydroxymethyl)-4-methoxyphenyl]-3,5-dimethyl-1H-pyrazol-4-yl}propanoic acid
7-(2,2-dimethylpropyl)-2-[3-(2-fluorophenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(2-methoxyphenyl)-3-(1-{1-[1-(1-methylcyclopropyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
9-[2-(3,4-dimethylphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(1H-imidazol-1-yl)-1H-indole
1-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
4-{[4-(2,5-dioxo-4-propylimidazolidin-4-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-({[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)cyclohexan-1-ol
N2-(3-methylpyridin-4-yl)-N1-(thian-4-yl)ethane-1,2-diamine
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
8-(3-fluoropyridin-4-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]benzene-1-sulfonamide
1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
1-[(4-chlorophenyl)methyl]-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
2-[(3-methoxyphenyl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}morpholine
2-(4-cyclobutyl-1-cyclopentylpiperazin-2-yl)ethan-1-ol
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide