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[1-({[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)cyclopropyl]methanol
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(pyridin-3-yloxy)piperidin-1-yl]propan-1-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(2-hydroxyethyl)-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-[3-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
3-[4-(benzyloxy)phenyl]pyrazine-2-carbonitrile
2-[(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]-6-methylpyridine-3-carbonitrile
N-[3-(dimethylamino)propyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-[(4-{thieno[3,2-d]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-yl)amino]acetic acid
3-{1-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}pyridine
8-chloro-2-(furan-2-yl)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}quinoline-4-carboxamide
2-(5-{1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethyl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
3-cyano-5-fluoro-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide
2-(methylamino)-N-[1-(3-methylphenyl)piperidin-4-yl]-1,3-thiazole-4-carboxamide
N-[3-(1H-indol-2-yl)phenyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-3-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(2-chloro-4-fluorophenyl)ethan-1-one
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}methanesulfonamide
2-oxo-2-[3-(4-phenoxybenzoyl)piperidin-1-yl]-N-(propan-2-yl)acetamide
4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1λ6-thiane-1,1-dione
2-ethyl-5-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}[(4-fluorophenyl)methyl]methylamine
2-{3-oxo-9-[(2E)-3-phenylprop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
[(2-chloro-3,4-dimethoxyphenyl)methyl][(1,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
N-(1,2-oxazol-3-ylmethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-{4-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylacetamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
1-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}cyclopentane-1-carboxamide
1-(1H-pyrazol-3-ylmethyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
1-[(1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-(4-{[(furan-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-(oxan-4-yl)-3,4-dihydropyrimidin-4-one
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-6-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
N'-(2,5-dimethylphenyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]propanediamide
N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-2-(trifluoromethyl)benzamide
(4aS,8aR)-6-(1H-1,3-benzodiazol-2-ylmethyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
(3S,4R)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]azepan-3-amine
4-(4-fluorophenyl)-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-4-ol
1-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(propan-2-yl)urea
5-[(4-methylpiperazin-1-yl)methyl]-N-[2-(3-methylthiophen-2-yl)ethyl]furan-2-carboxamide
(3S)-3-benzyl-4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperazin-2-one
{[(1R,5S,6S)-3-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
7-[(2,3-dimethoxyphenyl)methyl]-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-benzyl-5-{[(4-fluorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-[(5-methylfuran-2-yl)methyl]piperidine
2-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methoxybenzamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-1H-1,2,4-triazole-5-carboxamide