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5-chloro-4,6-dimethyl-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
N-butyl-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
6-methoxy-N-methyl-N-[3-(oxolan-2-yl)propyl]pyrimidin-4-amine
N-[2-(piperidin-1-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
N-(propan-2-yl)-6-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridazin-3-amine
3-acetamido-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}benzamide
2-[methyl(2-phenylethyl)amino]-N-(pyrrolidin-3-yl)-2,3-dihydro-1H-indene-2-carboxamide
4-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine-1-carboxamide
3-{3-[3-(dimethyl-1,3-thiazol-5-yl)phenyl]-1H-pyrazol-1-yl}-1,1,1-trifluoropropan-2-ol
N-ethyl-8-methoxy-N-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-phenyl-1-(1H-pyrazole-3-carbonyl)azepane
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
1-[(3-methoxyphenyl)methyl]-4-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-2-one
3-(1-methyl-1H-pyrrol-2-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]urea
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
2-(6-hydroxypyridine-3-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
2-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-1,3-thiazol-4-yl)methanol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-(1H-imidazol-1-yl)acetamide
3-({2-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(4-ethoxyphenyl)methyl]-2-methyl-N-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{2-[(dimethylamino)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
(3aR,5R,6S,7aS)-2-(1,3,7-trimethyl-1H-indole-2-carbonyl)-octahydro-1H-isoindole-5,6-diol
2-(1-ethylpiperidin-4-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
5-fluoro-4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}quinazoline
1-(2-chlorophenyl)-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
4-(1-butyl-1H-imidazol-2-yl)-1-(3,4-dimethylbenzoyl)piperidine
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-decahydro-2,7-naphthyridine-2-sulfonamide
1-[3-(2-{[(cyclobutylmethyl)(methyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
2-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-(butan-2-yl)-N-(pyridin-3-ylmethyl)isoquinoline-5-carboxamide
1-(4-chlorophenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]cyclopropane-1-carboxamide
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-[({1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
1-(2-methoxyphenyl)-3-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
[(5-chlorothiophen-2-yl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
(1S,4S)-2-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-2-azabicyclo[2.2.1]heptane
3-{[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzonitrile
2-{2-[3-(azocan-1-yl)propanamido]ethyl}-1,3-thiazole-4-carboxylic acid
3-[(4-fluorophenyl)formamido]-N-(1-propylpiperidin-4-yl)propanamide
(1-{[1-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
7-fluoro-3-{[methyl({2-[2-(prop-2-en-1-yl)phenoxy]ethyl})amino]methyl}-1,2-dihydroquinolin-2-one
N-ethyl-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
N-[(2,4-dimethoxyphenyl)methyl]-2-(4H-1,2,4-triazol-4-yl)benzamide
N-ethyl-3,4,5-trimethoxy-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide