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N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(2-ethylpyrimidin-5-yl)-6-fluoroquinoline
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-{pyrazolo[1,5-a]pyridin-7-yl}benzoic acid
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[(phenylcarbamoyl)carbonyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
3-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
2-{4-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}acetic acid
1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-4-(piperidin-1-yl)butan-1-one
3-(2H-1,3-benzodioxol-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{4-[3-(azetidine-1-carbonyl)benzenesulfonyl]-1-methylpiperazin-2-yl}methanol
2-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyridine-3-carboxamide
8-(2,1,3-benzothiadiazol-5-ylmethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[5-(2,3-dimethoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-{4-[4-(5,6-dimethylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]piperidin-1-yl}ethan-1-one
2-{3-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenoxy}acetamide
5-({[(4-fluorophenyl)methyl](prop-2-en-1-yl)amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
3-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-(4-oxo-4H-chromen-6-yl)urea
N-cyclohexyl-3-[(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)formamido]propanamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
1,9-dimethyl-4-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(dimethylamino)-3-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}propan-2-ol
3-methyl-1-(2-methylpropyl)-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-one
N-({5-[(2-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,5-dimethylfuran-3-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)methylamine
N-butyl-4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
2-(2-fluorophenoxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(2-aminoethyl)-N-[2-(azepan-1-yl)ethyl]quinazolin-4-amine
(2S)-2-acetamido-3-(1H-imidazol-4-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxypropyl)acetamide
(2S)-2-{4-oxo-3H,4H-pyrido[2,3-d]pyrimidin-3-yl}-3-phenylpropanamide
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrazolo[1,5-a]pyridine-7-carboxamide
1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
(3S,4S)-1-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-4-methylpiperidine-3,4-diol
8-(2-methoxyacetyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 2-[4-({[2-(2-oxopiperidin-1-yl)ethyl]carbamoyl}amino)phenyl]acetate
2-(4-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
2-[({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-4-carbonitrile
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-4-cyclobutaneamidobenzamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(pyridin-2-yl)propyl]-1,2-oxazole-3-carboxamide
N-[4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]acetamide
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-4-methylpiperidine-4-carboxamide
1-{3-[({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]propyl}pyrrolidin-2-one
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
1-(cyclobutylmethyl)-3-{[cyclohexyl(methyl)amino]methyl}-3-hydroxypiperidin-2-one
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[3-(1H-imidazol-5-yl)phenyl]urea
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
N'1-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}cyclopropane-1,1-dicarboxamide