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1-{3-[3-(methanesulfonylmethyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidin-3-ol
3-{[2-amino-6-(diethylamino)pyrimidin-4-yl]amino}propane-1,2-diol
2-[1-benzyl-5-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1H-1,2,4-triazol-3-yl]acetamide
1-(2-methoxyethyl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
1-ethyl-N-[3-(4-methoxyphenyl)propyl]-5-oxopyrrolidine-3-carboxamide
N-[1-(3-hydroxyadamantan-1-yl)ethyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-phenylethane-1,2-dione
N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
2-(2-fluoro-6-methoxyphenyl)quinoline
N-[3-chloro-4-(ethylcarbamoyl)phenyl]-3-hydroxy-3-phenylpyrrolidine-1-carboxamide
N-(pyridin-3-ylmethyl)-4-(thiophen-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(azepane-1-carbonyl)-1-propyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(butylsulfanyl)-N4-[(1,4-dimethylpiperazin-2-yl)methyl]pyrimidine-4,6-diamine
(4aS,7aR)-1-[(7-hydroxyquinolin-3-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}urea
3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2,6-dimethylquinoline
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-3-phenoxypropan-1-one
N4-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}pyrimidine-2,4-diamine
5,6-dimethoxy-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-dihydroisoquinolin-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(furan-2-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
methyl 4-[({2-[5-oxo-1-(oxolan-2-ylmethyl)pyrrolidin-2-yl]ethyl}amino)methyl]benzoate
2-[4-(4-cyclohexylpiperazine-1-carbonyl)-5-(propan-2-yl)-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
2-cyclobutanecarbonyl-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-[(3R,4S)-1-(1-benzothiophene-2-sulfonyl)-4-(dimethylamino)piperidin-3-yl]propanoic acid
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-(furan-2-ylmethyl)piperidin-4-amine
(4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}morpholin-3-yl)methanol
4-(2-methyl-4-phenylpyridine-3-carbonyl)-1,4-oxazepan-6-ol
2-{[7-(2,3-dihydro-1-benzofuran-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
methyl 2-(azocane-1-sulfonyl)-6-(1-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
N-[2-(2,6-dimethoxyphenoxy)ethyl]-1-oxaspiro[4.4]nonan-3-amine
4-{[1-(carbamoylmethyl)piperidin-4-yl]oxy}-3-chloro-N-(2-methoxyethyl)benzamide
6-methyl-2-({1-[3-(3-methylphenoxy)azetidin-1-yl]-1-oxopropan-2-yl}sulfanyl)-3,4-dihydropyrimidin-4-one
1-cyclohexyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
1-cyclopentyl-N-(3-methylbutyl)-4-oxo-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-methyl-N-[3-(methylsulfanyl)propyl]-1H-1,3-benzodiazole-5-carboxamide
9-benzoyl-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
2-(acetamidomethyl)-N-(4-fluorophenyl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
N-methyl-1-(6-methyl-2-propylpyrimidin-4-yl)-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
1-amino-N-{2-[1-(1-benzofuran-5-ylmethyl)piperidin-3-yl]ethyl}cyclopropane-1-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
(2R,6R)-10-methoxy-4-[2-(propan-2-ylsulfanyl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-methylpyridin-4-yl)piperazine
5-[(4-methoxynaphthalen-1-yl)methyl]-5-(3-oxo-3-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}propyl)pyrrolidin-2-one
4-{[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(2R,6R)-11-methoxy-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methoxybenzamide