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1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
N-({1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
N-[(2S)-4-(methylsulfanyl)-1-oxo-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}butan-2-yl]acetamide
8-(1H-imidazol-4-ylmethyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(1,4-dithiepan-6-yl)amino]-1-propylpyrrolidin-2-one
3-(2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}acetamido)propanoic acid
1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
(2S)-3-(4-hydroxyphenyl)-2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propanamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2H-1,3-benzodioxole-5-carboxamide
1-[(2-chlorophenyl)methyl]-4-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
(4aS,7aR)-1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3,4-difluorophenyl)methyl]-3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
[(2,3-dimethoxyphenyl)methyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-[(5-chlorothiophen-2-yl)methyl]-2-(3-methoxyphenyl)acetamide
3-(2-ethylbutyl)-8-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]naphthalene-2-sulfonamide
3-(5-chloro-2-methoxyphenyl)-1-[1-(furan-2-carbonyl)piperidin-3-yl]urea
N-(1-carbamoylcyclopentyl)-2-methyl-4-phenylpyrimidine-5-carboxamide
8-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{2,8-diazaspiro[4.5]decan-2-ylmethyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-[5-({[(2,5-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
5-(3,4-difluorophenoxymethyl)-N-(1-phenylcyclopropyl)-1,2-oxazole-3-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-{1-oxaspiro[4.5]decan-3-yl}propanamide
4-(6-ethylpyrimidin-4-yl)-N-(4-oxo-4H-chromen-6-yl)piperazine-1-carboxamide
2,7,8-trimethyl-4-[2-(pyridin-2-yl)piperidine-1-carbonyl]quinoline
2-methoxy-5-({[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]carbamoyl}amino)benzamide
1-(2-methylphenyl)-N-[2-(4-methylpiperazin-1-yl)butyl]piperidin-4-amine
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidine
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl][2-methyl-2-(morpholin-4-yl)propyl]amine
N-[2-(methylsulfanyl)ethyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
N-ethyl-3-(4-methylphenyl)-3-phenyl-N-(pyridin-4-ylmethyl)propanamide
4-chloro-N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-[2-(hydroxymethyl)phenyl]-1,2-dihydroquinolin-2-one
N,N,5,7-tetramethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
1-{imidazo[1,2-a]pyridine-3-carbonyl}-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)acetamide
2-[4-({2-[6-(dimethylamino)pyridin-3-yl]-1H-imidazol-1-yl}methyl)piperidin-1-yl]ethan-1-ol
(1,3-benzothiazol-2-ylmethyl)({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-4-hydroxy-2-methylpyrimidine-5-carboxamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
{[(3S,4R)-1-[2-(4-fluorophenoxy)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-(prop-2-en-1-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-[(oxan-4-ylmethyl)amino]pyridine-3-carboxamide
N-(thiophen-2-ylmethyl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
6-[(2-{4-[(dimethylamino)methyl]thiophen-2-yl}-1H-imidazol-1-yl)methyl]pyrimidin-4-ol
4-(4-methylpyrimidin-2-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cyclohexyl-4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepane