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7-[(3,4-difluorophenyl)methyl]-2-(3-ethynylbenzoyl)-2,7-diazaspiro[4.5]decane
2-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]naphthalen-1-ol
3-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
(3S,4R)-1-cyclopentanecarbonyl-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}-4-methyl-1H-1,3-benzodiazole
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,7,8-trimethylquinoline-4-carboxamide
2-(phenylsulfanyl)-1-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-methyl-N-(3-{[(2-methylphenyl)methyl]sulfanyl}propyl)-5-oxopyrrolidine-3-carboxamide
2-amino-3-ethyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}phenyl)-1H-imidazole
4-[5-(cyclopropylmethyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
1-[9-hydroxy-7-(thianthren-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
1-(4-fluorophenyl)-4-[1-(propan-2-yl)piperidine-3-carbonyl]-1,4-diazepane
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(prop-2-en-1-yloxy)benzoyl]-decahydro-1,6-naphthyridin-2-one
3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(2H-1,3-benzodioxol-5-yl)acetamide
N,2-dimethyl-N-(1-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)furan-3-carboxamide
(3R,4S)-1-[2-methoxy-5-(1,2-oxazol-5-yl)benzenesulfonyl]-4-propylpyrrolidin-3-amine
3-[1-(2-methoxyethyl)-2-methyl-1H-indol-5-yl]-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
(1S,5R)-3-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(dimethylamino)-4-methyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
N-(4-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}phenyl)acetamide
4-(4-methoxyphenyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
1-(2-methoxybenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
3-[3-(4-chlorophenyl)phenyl]-1-methyl-1-(oxan-4-yl)urea
1-(4,6-dimethylquinazolin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]piperidine-4-carboxamide
(1R,5R)-6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]pyridine-3-carbonitrile
2-{4-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
1-ethyl-3-(2-methylpropyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
(3aS,6aS)-5-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-(1-cyclopentyl-4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(pyridin-2-yl)ethyl]acetamide
4-(5-methyl-1,3-oxazole-4-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-benzyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N,4-dimethyl-N-(pyridin-3-ylmethyl)-6H,7H,8H-cyclopenta[g]quinazolin-2-amine
4-({[4-methyl-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)pyridine
(3S)-1-(1H-indol-5-ylmethyl)-N,N-dimethylazepan-3-amine
(3S,4S)-1-[6-(dimethylamino)pyridine-3-carbonyl]-4-propylpyrrolidine-3-carboxylic acid
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazine
(4aR,8aR)-4a-hydroxy-7-[(2-methoxy-4-methylphenyl)methyl]-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
4-(3,4-difluorobenzoyl)-1-(4-methylphenyl)piperazin-2-one
5-(1-benzylpiperidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
1-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-4-(3-methylpyridin-2-yl)piperazine
(3S,4R)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
7-(2-hydroxyethyl)-2-{2-[2-(trifluoromethyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
3-(3,4-dimethoxyphenyl)-5-{1-[2-(furan-3-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole