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2-(5-{[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]methyl}-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl)pyridine
(3R,4R)-1-[(2-ethylpyrimidin-5-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3,3-diphenylpropanamide
2-(adamantan-1-yl)-4-hydroxy-N-(3-hydroxy-3-methylbutyl)-N-methylpyrimidine-5-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[4-(furan-2-yl)pyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
(1S,5R)-6-benzyl-3-[2-(4-methoxyphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-hydroxy-3-methylbutyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
(2S)-N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-2-(methoxymethyl)pyrrolidine-1-carboxamide
1-ethyl-4-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)pyrrolidin-2-one
4-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl}benzoic acid
N-(2,4-dimethylphenyl)-3-{6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-3-oxopropanamide
2-{[4-(2-chlorophenyl)-5-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
methyl 8-{[4-(methoxycarbonyl)phenyl]methyl}-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[4-(methylsulfanyl)phenyl]-1H-imidazole
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-(cyclohexylmethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[1-(3-phenylpropyl)-4-(pyridin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
3-(cyclopropylmethyl)-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethyl-4-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1,3-oxazole-5-carboxamide
1-[2-(4-fluorophenyl)ethyl]-4-[(1-methylpiperidin-4-yl)amino]pyrrolidin-2-one
N-[2-(1,3-benzoxazol-2-ylsulfanyl)ethyl]-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
2-{4-[(5-cyclopentylthiophen-2-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(thiophen-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
5-(azepane-1-carbonyl)-N-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-benzotriazole
2-[5-(2,3-dihydro-1H-inden-2-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[3-(2,3-dichlorophenyl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
N-[2-(1H-indol-1-yl)ethyl]-1-methanesulfonyl-N-methylpiperidin-4-amine
2-(3-chloro-4-methoxyphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
(1S,9S)-11-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-{[(3S,4S)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-1-yl]methyl}quinolin-4-ol
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-(oxan-2-ylmethyl)acetamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
(3R)-3-hydroxy-N-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
1-[(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]-2-methyl-1H-1,3-benzodiazole
3-[(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)amino]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
5-chloro-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,2-dimethylpyrimidine-4-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{2-[1-(2-hydroxy-2-phenylacetyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
2-{1-[(4-fluorophenyl)methyl]-4-propylpiperazin-2-yl}ethan-1-ol
(E)-N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-2-phenylethene-1-sulfonamide
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
N-[(3-methyloxetan-3-yl)methyl]-3-phenylbenzamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one