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1-(4-{2-[(4aR,8aS)-6-(4-phenylbutanoyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
(3aS,6aS)-2-ethyl-5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-benzylpiperidin-4-yl)-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(2-methoxyphenyl)piperazin-1-yl]propan-1-one
N-{3-[methyl(phenyl)amino]propyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
6-[(diethylamino)methyl]-N-(3,5-dimethylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{4-[(3-methylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-{6-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]pyridin-3-yl}ethan-1-one
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-(4-fluoro-2-methylbenzoyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
5-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)pyrazin-2-ol
3-[(2R,3R,6R)-5-[(5-ethylpyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
5-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
1-methyl-N-(quinolin-3-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
7-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
1-(pyridin-3-ylmethyl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
2-{4-[3-(2-methylpropyl)morpholine-4-carbonyl]phenoxy}-1-(piperidin-1-yl)ethan-1-one
1-(carbamoylmethyl)-N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxamide
1-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)-2-(pyridin-2-yl)ethan-1-one
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-methyl-N-{3-oxo-3-[4-(2-phenylethyl)piperidin-1-yl]propyl}methanesulfonamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,4-diazepan-5-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpropanamide
4-[1-(pyridin-3-yl)-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethyl]morpholine
3-({1-[3-(3-chlorophenyl)phenyl]piperidin-4-yl}amino)propanamide
N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
2-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine-3-carbonyl]pyridine
ethyl 1-(2-methylfuran-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
3-(4-methoxyphenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-phenylpropanamide
4-{5-[2-(oxolan-2-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl}pyridine
ethyl 1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
8-{furo[3,2-c]pyridin-4-yl}-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-ethyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(2,2,2-trifluoroethyl)acetamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,4-diazepane-6-carboxylic acid
2-chloro-N-{[1-(propane-1-sulfonyl)piperidin-3-yl]methyl}benzamide
(2S)-2-amino-3-(1H-indol-3-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
7-fluoro-2-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-3-methyl-1H-indole
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
N,N-diethyl-5,7-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-[(2S,4R,6R)-2-(3-acetylphenyl)-6-(propan-2-yl)oxan-4-yl]acetamide
7-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine