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1-(4-phenyl-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)ethan-1-one
1-(4-aminopyrimidin-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(3-methylbut-2-enoyl)pyrrolidine-3-carboxylic acid
3-phenyl-5-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
(4S)-4-(propan-2-yl)-3-{[4-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
(2-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-1,3-thiazol-4-yl)methanol
4-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]morpholine
(3R,4S)-4-cyclopropyl-1-(1-phenylcyclopentanecarbonyl)pyrrolidin-3-amine
N-[2-(2,3-dichlorophenyl)ethyl]-2-ethylpyrimidine-5-carboxamide
2-(2-phenylethyl)-9-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-[1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(3-benzyl-1H-1,2,4-triazol-5-yl)phenyl]acetamide
2-({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-[1-(1H-indol-2-ylmethyl)-3-oxopiperazin-2-yl]-N-methylacetamide
methyl 4-(5-{[2-(2-ethoxy-2-oxoethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
8-[1-(4-methylphenyl)cyclopropanecarbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(2,3-difluoro-4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
8-(4,6-dimethoxypyrimidin-2-yl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1H-indol-3-yl)-1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
6-tert-butyl-N-(1-methoxybutan-2-yl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(3-methoxyphenyl)-N-methylacetamide
6-(4-fluorophenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-phenoxy-1-[4-(pyrazin-2-yl)piperazin-1-yl]butan-1-one
2-(prop-2-en-1-yl)-9-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(1H-imidazol-5-yl)ethyl]-3-(2-methoxyethyl)-5-(2-methyloxolan-2-yl)-1H-1,2,4-triazole
ethyl 3-[(3-methoxyphenyl)methyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxylate
6-[(diethylamino)methyl]-N-(quinolin-8-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(2-methylpyrimidin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{3-[(benzyloxy)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-ethyl-1,2-oxazole
(1R,5S,6R,7S)-6-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-3-methyl-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-methyl-N-(oxolan-2-ylmethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
N-(2-methoxyethyl)-3,4,7-trimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
5-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2,1,3-benzothiadiazole
N-[3-(4-{[(3-ethyl-5-methyl-1,2-oxazol-4-yl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
3-chloro-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
4-(cyclohexylmethyl)-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
1-[2-(methylsulfanyl)ethyl]-4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperazine
4-{4-[(4-methoxynaphthalen-1-yl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(5-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1H-1,2,4-triazol-1-yl)butan-2-ol
4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-oxo-1-phenyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,5-dihydro-1H-pyrazole-3-carboxamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
5-({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(3,5-dimethylphenyl)-N-(1,3-thiazol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine