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5-butyl-1'-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,3s,6r,8S)-4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
[(3R,4R)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
4-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]thiomorpholine
7-(cyclopropylmethyl)-N-(2-fluoroethyl)-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-cyano-N-{1-[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}benzamide
1-[1-(ethanesulfonyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-[5-(1-acetylpiperidin-4-yl)-1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
(1R,5R)-3-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-azabicyclo[3.3.1]nonane
9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-2-(pyridin-4-yl)acetamide
1-(5-methoxyfuran-2-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
2-(1-benzyl-4-cyclobutylpiperazin-2-yl)ethan-1-ol
2-phenyl-1-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]ethan-1-one
dimethyl({[4-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-2-yl)phenyl]methyl})amine
[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-(cyclopropylmethyl)-6-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-5-methoxy-1-methyl-1H-indole
(3aS,6aS)-5-(isoquinolin-1-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methoxy-1-{4-[4-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
ethyl 4-{2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
3-(2,3-dihydro-1H-inden-5-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]urea
4-[3-(dimethylamino)benzoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
2-[methyl({4-methyl-5-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
(1S,5R)-N-[4-(dimethylamino)phenyl]-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
[(2S,6S)-4-(2-methylfuran-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
3-benzyl-4-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
N,2,6-trimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyrimidine-4-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
4-methyl-5-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
3-[2-({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyridin-3-yloxy)ethyl]azepan-4-amine
2-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-1,8-naphthyridine
3-(4-fluorophenyl)-N-[2-(methylamino)ethyl]-3-phenylpropanamide
3-cyano-N-(2-ethyl-3-methyl-1-benzofuran-7-yl)piperidine-1-carboxamide
N-ethyl-1-methyl-3-phenyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
5-methyl-N-({3-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
(2-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-yl)methanol
5-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
(1S,4S)-2-(3-chlorophenyl)-5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
1-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-4-(azepan-1-yl)butane-1,4-dione
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-(cyclohexylmethyl)-4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1H-indole-6-carboxamide