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[1-(2-methyl-1H-imidazol-1-yl)propan-2-yl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
5-(methoxymethyl)-N-[(4-methoxyphenyl)methyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
[1-(pyrazin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(2E)-3-phenylprop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
4-(2-amino-3-cyano-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl)-N-methylbenzene-1-sulfonamide
2-(4-cyclohexylphenyl)-5-(methanesulfonylmethyl)pyridine
N3-cyclohexyl-1-(2-methoxyethyl)-N3-methyl-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-methyl-6-[4-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
N-{2-[3-(trifluoromethyl)phenyl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[3-(3-methylphenyl)phenyl]-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-3-carboxamide
4-(1,3-benzothiazol-2-yl)-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(5-chlorothiophen-2-yl)methyl]-3-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]urea
2-chloro-N-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(pyridin-2-ylmethyl)acetamide
1-[5-(ethanesulfonyl)thiophen-2-yl]-4-phenyl-1H-imidazole
1-methyl-4-(4-phenoxybutyl)-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
5-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(4-fluorophenyl)methyl]-2-(2-methoxyacetamido)-N-(prop-2-en-1-yl)benzamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[2-(dimethylamino)ethyl]-N-[2-(naphthalen-1-yl)propan-2-yl]-5-oxopyrrolidine-3-carboxamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-cyclopentylacetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
4-[(4-methoxyphenyl)methyl]-1-(9-methyl-9H-carbazole-3-carbonyl)-1,4-diazepan-5-one
(1S,5R)-3-benzyl-6-(2-propyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[6-(thiomorpholin-4-yl)pyridazin-3-yl]benzoic acid
3-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopent-3-en-1-amine
1-(2-ethoxyethyl)-5-(3,3,4-trimethylpiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(1H-imidazol-1-ylmethyl)-1-(1,3-thiazol-2-ylmethyl)piperidine
4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidine
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
7-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decane
N-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(2-phenylethyl)propanamide
1-[4-(furan-2-yl)benzoyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
(1S,5R)-3-(4-methylpiperidine-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1S,2R)-2-aminocyclobutyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(3-phenylpropanoyl)piperidin-4-yl]propanamide
8-[2-(2-oxopyrrolidin-1-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-5-(morpholin-4-ylmethyl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]furan-3-carboxamide
2-(cyclopropylmethyl)-9-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
(3aR,6aR)-2-cyclobutanecarbonyl-5-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
N-(3,4-difluorophenyl)-6-(2-methoxybenzoyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methylpyridine-3-carboxamide
2-amino-6-benzyl-4-(furan-2-yl)-8-methyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}butane-1,2-dione
(4aS,7aR)-1-(furan-3-ylmethyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-(propan-2-yl)pyridine-4-carboxamide