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N-methyl-N-[1-({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)pyrrolidin-3-yl]acetamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
1-[5-(azepan-1-ylmethyl)-2-methoxyphenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
4-{2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carbonyl}-1-(4-methylphenyl)piperazin-2-one
N3-ethyl-N1-[2-(2-methoxyphenoxy)phenyl]pyrrolidine-1,3-dicarboxamide
1-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
3-{2-[4-(3,5-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
(2S)-1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-methyl-2-(propan-2-yl)piperazine
(1R,6S)-N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
4-(2,5-dimethylthiophen-3-yl)-2-[4-(2-ethylpiperidine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]pyrimidine
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
4-(2-fluoro-5-methylphenoxy)-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxylic acid
[(3-methoxyphenyl)methyl](prop-2-en-1-yl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
3-{[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]methyl}pyrrolidin-3-ol
4-(hydroxymethyl)-1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
1-(cyclohexylmethyl)-N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-(3-methyl-1H-1,2,4-triazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-({1-[4-(propan-2-yl)phenyl]-1H-pyrazol-4-yl}methyl)pyrrolidin-3-ol
methyl (2S)-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-2-phenylacetate
2-(4-chloro-1H-pyrazol-1-yl)-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-{3-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]phenyl}ethan-1-amine
4-[(4-methoxy-2,5-dimethylphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1R,3S)-N-[(2,4-dichlorophenyl)methyl]-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carboxamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(3-hydroxypropyl)-N-(propan-2-yl)benzamide
2-(cyclopropylmethyl)-9-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(5-propyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-methoxyethyl)-1-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
6-(2-chlorobenzoyl)-1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octane
(1R,5R)-3-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-3,9-diazabicyclo[3.3.2]decan-10-one
N-{4-[4-(2-oxopyrrolidin-1-yl)butanamido]phenyl}pentanamide
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,6R)-9-{1-[(4-methoxyphenyl)amino]cyclopentanecarbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-{[(cyclobutylmethyl)(oxolan-2-ylmethyl)carbamoyl]amino}-2-methoxy-N,N-dimethylbenzamide
3-(2-hydroxyphenyl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrazole-5-carboxamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-5-carboxamide
N-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
2-(3-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
3-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-N-(2,3-dihydro-1H-inden-5-yl)-5-(methylsulfamoyl)benzamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(oxane-4-carbonyl)piperidine-4-carboxylic acid
1-[(4-methoxypyridin-2-yl)methyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-sulfamoylbutanamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(2-hydroxyphenyl)acetamide
5-{[(3-cyclopentylpropyl)(methyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]-3-propyl-1H-pyrazole-5-carboxamide
4-(furan-2-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-benzyl-1-(4-methylphenyl)-4-(1,2-oxazole-3-carbonyl)piperazin-2-one
4-(1H-imidazol-2-ylmethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)quinazoline