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1-{1'-[3-(dimethylamino)pyrazin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
1-[1-(4-benzylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]-2-(thiophen-3-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(2-ethyl-1H-imidazol-1-yl)propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,5-dimethylfuran-3-carboxamide
2-(4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)ethan-1-amine
2-(2,3-dihydro-1H-isoindol-2-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-dimethoxyphenyl)acetamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
1'-[(2-fluoro-4-methoxyphenyl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(2-methylphenyl)-1,4-diazepane
1-{4-hydroxy-2-[(phenylsulfanyl)methyl]pyrimidine-5-carbonyl}piperidine-3-carbonitrile
1-[1'-(5-methyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
(2S)-N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)oxolane-2-carboxamide
4-{1-methyl-5-[pyridin-3-yl(pyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-3-yl}benzamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
1-(5-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
4-({2-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
ethyl 1-{1-[6-(dimethylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}piperidine-4-carboxylate
4-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)pyridine
ethyl 3-[(3-chlorophenyl)methyl]-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine-3-carboxylate
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-methyl-N-(pyridin-4-ylmethyl)-1H-pyrrole-3-carboxamide
N-cyclohexyl-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
1-[(1-{6-[(cyclopropylmethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]piperidin-4-ol
(1R,3S,5S)-8-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-8-azabicyclo[3.2.1]octan-3-ol
1-(3-chlorophenyl)-5-methyl-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one
N-(furan-3-ylmethyl)-N-methyl-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-phenoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-N-[2-(3-chlorophenyl)ethyl]-4-(2-methoxyacetamido)-1-methylpyrrolidine-2-carboxamide
1-butyl-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H,4H-pyrazolo[3,4-d]imidazole
(3R,4S)-4-(5-methylfuran-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]pyrrolidin-3-amine
1-butyl-3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]urea
7-cyclopentyl-2-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-(2-chlorophenyl)-2-methyl-N-[2-(pyridin-2-yl)ethyl]furan-3-carboxamide
N-(3,4-dimethoxyphenyl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
3-[2-(5-chloro-2,4-dimethoxyphenyl)-1H-imidazol-1-yl]-1,1,1-trifluoropropan-2-ol
(1S,9aR)-1-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-octahydro-1H-quinolizine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methoxypyridine
1-(1-benzylpiperidin-4-yl)-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
6-methyl-N-(3-phenylprop-2-yn-1-yl)-N-propylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[3-(2,6-dimethylphenoxy)azetidin-1-yl]propane-1,3-diol
1-(cyclopropanesulfonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}acetic acid
2-amino-6-(4-chloro-3-methylphenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
1-methyl-3-(piperidine-1-carbonyl)-N-[(3,4,5-trimethoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine