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7-ethyl-1-[2-(4-fluorophenyl)morpholine-4-carbonyl]-3-methyl-5H,6H,7H,8H-imidazo[1,5-a]pyrazin-8-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
{5-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1,3-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(2-methylpropyl)piperidin-4-amine
N-cyclopropyl-3-[5-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
5-{[benzyl(methyl)amino]methyl}-N-(1H-indol-6-ylmethyl)-1,2-oxazole-3-carboxamide
(3R,4R)-4-(morpholin-4-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-ol
7-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)piperidin-2-one
4-(furan-2-ylmethyl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
9-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-(4-methyl-1H-pyrazol-1-yl)-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-N'-phenylethanediamide
(3S,4S)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
(4aR,7aS)-N,N-dimethyl-4-[(4-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-amino-4-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidine-5-carboxamide
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
2-[2-(2,4-dimethoxyphenyl)phenoxy]propanamide
6-[(3S)-1-benzylpiperidin-3-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-5-(methoxymethyl)furan-2-carboxamide
2-{1-[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,3-benzodiazole
1-[2-(2-methoxyphenyl)ethyl]-5-(oxan-4-yl)-4-phenyl-1H-imidazole
3,6-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-N-(propan-2-yl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
1-{5-[(4,4-difluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
(2R)-2-[(2-amino-5-ethylpyrimidin-4-yl)amino]-2-phenylethan-1-ol
ethyl 4-[2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]piperazine-1-carboxylate
6-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-9H-purine
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
6-(5-chloro-2-ethoxyphenyl)-N-methylpyridine-2-carboxamide
3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
5-[5-(1H-imidazol-1-ylmethyl)furan-2-yl]-3-(oxan-4-yl)-1H-1,2,4-triazole
methyl 1-[(3R,5S)-1-[(2-methoxyphenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
[(3-chloro-5-fluorophenyl)methyl](methyl){[1-(propan-2-yl)piperidin-3-yl]methyl}amine
6-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}pyridine-2-carboxylic acid
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
1-(4-benzylpiperazin-1-yl)-3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-3-yl]propan-1-one
N-(2-hydroxyethyl)-3-[5-(oxan-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
3-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-6-methyl-2-[(2-methylphenyl)methyl]-1-(pyridin-4-ylmethyl)-1,4-dihydropyridin-4-one
1-(5-acetyl-2-methoxyphenyl)-3-(2,2,2-trifluoroethyl)urea
2-{1-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-3-yl}-1H-1,3-benzodiazole
(2R,3R,6R)-3-(4-methylphenyl)-5-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1-phenylethyl)benzamide
3-{5-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5-fluoro-1H-1,3-benzodiazole
methyl (2R)-2-{[2-(4-methoxyphenoxymethyl)-1,3-oxazol-4-yl]formamido}propanoate
N-methyl-N-[1-(1-{[(pyrazin-2-yl)carbamoyl]methyl}-1,2,3,6-tetrahydropyridin-4-yl)ethyl]acetamide