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N4-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-3-(2-methylphenyl)-1,2,4-oxadiazole
(2R,3S)-2-{[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}-3-hydroxybutanoic acid
N-(furan-2-ylmethyl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-methyl-4-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
[(3R,4R)-1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-phenylpropan-1-one
N-{3-[({3-[(5-methylpyridin-2-yl)amino]propyl}carbamoyl)methoxy]phenyl}propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-methoxyfuran-2-carbonyl)piperidin-3-ol
N-({4-[(dimethylamino)methyl]phenyl}methyl)-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(cyclopropylmethyl)-4-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperazine
methyl (2S,4S)-1-methyl-4-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamido]pyrrolidine-2-carboxylate
(1S,5R)-3-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
[2-ethoxy-5-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenyl]methanol
ethyl 4-{2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamido}piperidine-1-carboxylate
5-methoxy-N,1-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-indole-2-carboxamide
1-(4-phenylpiperazine-1-carbonyl)-6-propyl-6-azaspiro[2.5]octane
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-3-[methyl(1-methylpyrrolidin-3-yl)sulfamoyl]benzamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl){[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}amine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
5-(2-chloro-4-methoxyphenoxymethyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1H-pyrazole
1-({1-[(2-chloro-4,6-dimethoxyphenyl)methyl]piperidin-3-yl}methyl)pyrrolidin-2-one
4-(3-chloro-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}phenyl)-4H-1,2,4-triazole
1-(but-2-ynoyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-cyclopentyl-N-(6-methylpyridin-3-yl)-6-oxopiperidine-3-carboxamide
5-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-2-yl}-2-(2-methylphenyl)pyrimidine
2-cyclohexyl-1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
1-[(2-carboxythiophen-3-yl)sulfonyl]-3-propylpiperidine-3-carboxylic acid
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(propylsulfanyl)acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(piperidin-4-ylmethyl)benzamide
5-({[4-(2,4-dioxoimidazolidin-1-yl)phenyl]formamido}methyl)-N-methylfuran-2-carboxamide
3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-2H-chromen-2-one
(4-{[3-(trifluoromethyl)phenyl]methyl}-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-4-yl)methanol
3-chloro-4-[(1-cyclopentanecarbonylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(thiophen-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(1-methylcyclopropyl)pyridine-3-carbonitrile
2-[({[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}amino)methyl]-5,8-dimethylquinolin-4-ol
1-(piperidine-1-sulfonyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-cyclohexyl-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-benzoxazole-6-carboxamide
9-(2,2-dimethyl-1-phenylcyclopropanecarbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-amino-4-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]propan-1-one
8-(2-aminopyridine-4-carbonyl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(4-methoxyphenyl)-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H-pyrazole-5-carboxamide
(4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}morpholin-2-yl)methanamine
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea