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1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-cyclopropyl-2-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]pyridine-4-carboxamide
N-{2-[2-(3-fluorophenyl)-6-oxo-1,6-dihydropyrimidin-4-yl]ethyl}-2-(furan-2-yl)-2-oxoacetamide
methyl 8-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1,2-dimethyl-3-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-1H-indol-5-ol
4-[(1-{[1-(2-fluorobenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-{6-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
1-[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]-N-methylcyclohexane-1-carboxamide
1-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}piperidine-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
3-acetamido-N-methyl-N-[3-(pyrrolidin-1-yl)butyl]benzamide
N-benzyl{[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]amino}sulfonamide
3-cyano-N-[(1R,3S)-3-(4-ethoxypiperidine-1-carbonyl)cyclopentyl]-5-fluorobenzamide
9-(morpholine-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{2-[3-(carboxymethyl)pyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-[3-methyl-4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]methanesulfonamide
N-[(3R,4S)-1-(1,3-dihydroxypropan-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-ol
5-(2-fluoro-6-methoxyphenyl)-1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazole
{1-[(1-methyl-1H-indol-5-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
N-(furan-2-ylmethyl)-2-[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxane-4-carboxamide
1,9-dimethyl-N-[3-(methylsulfanyl)phenyl]-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
N-[3-(1H-indazol-1-yl)propyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
(3aR,6aS)-2-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-5-methyl-octahydropyrrolo[3,4-c]pyrrole
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonitrile
1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-4-(2-methoxyphenyl)piperazine
1-cyclopentanecarbonyl-N-methyl-N-(1,2-oxazol-5-ylmethyl)piperidine-4-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(4-methyl-1H-pyrrole-2-carbonyl)morpholine
9-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
7,7-dimethyl-2-(1-methylpiperidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-amino-N-{[4-(aminomethyl)phenyl]methyl}-4-phenylpyrimidine-5-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-aminopiperidin-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
2-(5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-pyrazol-3-yl)pyridine
2-(1H-imidazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-cyclopropyl-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperazine-2-carboxamide
4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(2R)-3-(benzyloxy)-2-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
4-[(4-fluorophenyl)methyl]-1-(2-methoxy-2-methylpropanoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-(2,3-dihydro-1H-inden-2-yl)-N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)azepan-4-amine
2-(4-fluorophenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
1-[1-(pyridazine-3-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine