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3-{[(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
2-(2-chloro-4-fluorophenyl)-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(pyrimidin-2-ylmethyl)piperidin-3-yl]propanoic acid
N-methyl-2-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
2-{4-[1-ethyl-3-(4-fluorophenoxymethyl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
3-{1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-6-(3-methyl-3-phenylpiperidine-1-carbonyl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
(3S,4R)-1-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]benzamide
8-[(4-hydroxyphenyl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methylpropyl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{2-[4-(1H-pyrazol-5-yl)phenyl]quinolin-3-yl}methanol
1-(2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3-dihydro-1H-inden-2-yl)piperidine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-5-(methoxymethyl)-N-methylfuran-2-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}quinoxaline-5-carboxamide
6-fluoro-4-[3-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
8-(1H-1,3-benzodiazole-5-carbonyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,9aR)-8-benzyl-3-(hydroxymethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(furan-2-yl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-4-carboxamide
2-(propan-2-yl)-5-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1,3-benzoxazole
2-{5-[3-(piperidin-4-ylmethyl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
3-{[1-(oxolane-3-carbonyl)piperidin-4-yl]methyl}benzoic acid
(4aR,8aS)-6-[(4-hydroxy-3-methoxyphenyl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
2-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(4-fluorophenyl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]cyclopropane-1-carboxamide
(4aS,8aR)-2-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-decahydroisoquinoline
4-(azepane-1-carbonyl)-2-(1-tert-butyl-1H-pyrazol-4-yl)quinoline
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
1-cyclohexyl-3-methyl-5-[3-(pyrrolidin-1-yl)butyl]-1H-1,2,4-triazole
1-(2-aminoethyl)-N-[(4-chlorophenyl)(phenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
methyl (2S)-2-({1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-2-phenylacetate
2-methyl-3-oxo-N-[4-(propan-2-yl)phenyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
(1-{[2-(difluoromethoxy)phenyl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
4-{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}benzoic acid
1-[2-amino-6-(methylamino)pyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{1-benzyl-5-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
3-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}pyrrolidine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3,4,5-trimethoxy-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
1-(5-{[(furan-3-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol
5-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-hydroxy-N-[3-(2-methylpyrimidin-4-yl)phenyl]-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
1-(1-benzofuran-2-ylmethyl)-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
N-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylpyridine-2-carboxamide
2-(3-chlorophenoxy)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
2-(2-methyl-1H-imidazol-1-yl)-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one