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methyl 3-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
2-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]ethan-1-ol
4-phenyl-8-[2-(pyridin-3-yl)-1H-imidazol-1-yl]quinoline
5-chloro-N-[2-(2-fluorophenyl)-2-hydroxyethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-(5-propylthiophene-3-carbonyl)pyrrolidine-2-carboxamide
2-(1H-1,2,3,4-tetrazol-1-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
3-fluoro-N,7-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(3-methylphenoxy)piperidine
2-(dimethylamino)-2-(3-methylphenyl)-N-[3-(3-oxopiperazin-1-yl)propyl]acetamide
3-[(3R,4S)-1-[3-(2-methylphenyl)propanoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N,N-dimethyl-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-sulfonamide
N,2-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2R,6R)-6-methyl-1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
(1S,5R)-6-benzyl-3-(2-phenoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)-N-methylacetamide
(2S)-1-[(1-{[1-(pyridin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidine-2-carboxamide
methyl[(1-propyl-1H-imidazol-2-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-(2-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)piperidin-2-one
5-{6-methylimidazo[1,2-a]pyridin-2-yl}-3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4-fluoro-3-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]benzene-1-sulfonamide
2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]acetic acid
4-methyl-13-[4-(1H-pyrazol-1-yl)phenyl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
(1S,5R)-3-{2-methylthieno[2,3-d]pyrimidin-4-yl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[1-(dimethyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]methanol
6-ethyl-4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-(3-methoxyphenoxy)-1-(3-methylbutyl)azetidine
4-[1-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)piperidin-3-yl]benzoic acid
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-[(3S)-2-oxoazepan-3-yl]propanamide
5-cyclobutanecarbonyl-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[(3,5-difluorophenyl)methyl]-8-[3-(1H-imidazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
1-phenoxy-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propan-2-ol
N-[1-(3,5-difluorophenyl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-benzyl-3-hydroxy-N-(3-hydroxy-2-methylpropyl)pyridine-2-carboxamide
3,5-dimethyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]-1,2-oxazole-4-carboxamide
3-(2-fluorophenyl)-4-(1H-imidazol-2-yl)-1-methyl-1H-pyrazole
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-(4-phenylazepan-1-yl)propan-1-one
N-cyclopropyl-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
4-[(2-chlorophenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-methoxy-3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-[(2-chlorophenyl)methyl]-4-{3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-phenoxy-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-4-carboxylic acid
(4aR,7aS)-4-(1-benzofuran-2-ylmethyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(diethylamino)-3-(2-methoxy-4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(3R,4R)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-{[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylpyridin-2-amine