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4-chloro-3-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-5-amine
ethyl 4-{[1-(4-{[(2-fluorophenyl)methyl]carbamoyl}phenyl)piperidin-4-yl]amino}piperidine-1-carboxylate
4-[3-ethyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-N-methyl-1,3-thiazol-2-amine
1-(1-methylpiperidin-4-yl)-4-(1H-pyrazole-4-carbonyl)piperazine
N,N-dimethyl-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-[4-(4-amino-5-methylpyrimidin-2-yl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
methyl 2-{[(2-fluoro-6-methoxyphenyl)methyl]amino}pyridine-4-carboxylate
6-amino-2-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]pyrimidin-4-ol
N2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
1-[2-(quinolin-2-yl)phenyl]ethan-1-one
(2S,4R)-4-amino-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2-dihydroquinolin-2-one
2-{methyl[6-(6-methylquinolin-3-yl)pyridazin-3-yl]amino}ethan-1-ol
2-[4-(cyclopentylmethyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(1H-imidazol-2-ylmethyl)-N-methylpiperidin-3-amine
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amine
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-(pyrazin-2-yl)piperidin-3-amine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
2-{[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]amino}-2-(4-fluorophenyl)ethan-1-ol
N-[3-(4-methoxyphenyl)propyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
4-({[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]amino}methyl)-2,6-dimethylphenyl acetate
N-cycloheptyl-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine-4-carboxamide
methyl (2S,4S)-1-(1-methylpiperidin-4-yl)-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
1-ethyl-5-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-3-(propan-2-yl)-1H-pyrazole
1-[(2-chloro-6-fluorophenyl)methyl]-5-{[(cyclopropylmethyl)sulfanyl]methyl}-3-methyl-1H-1,2,4-triazole
N-{[4-(aminomethyl)phenyl]methyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-(2-{1-[2-(ethylsulfanyl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}piperidin-1-yl)ethan-1-one
(1S,9R)-11-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(1,4-oxazepan-6-ylmethyl)-3-(2,4,4-trimethylpentan-2-yl)urea
(3R,4R)-4-amino-1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-ol
4-methyl-5-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
2-{[1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-yl]oxy}pyrimidine
(2R,6S)-2,6-dimethyl-4-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)morpholine
1-(3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)-2-phenylethane-1,2-dione
1-(6-aminopyrimidin-4-yl)-4-(2H-1,3-benzodioxol-5-yloxy)piperidine-4-carboxylic acid
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
(2S,4R)-4-amino-1-(1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-N-ethylpyrrolidine-2-carboxamide
3-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
2-chloro-5-(2-ethoxypyridin-3-yl)pyrazine
2-(3-hydroxypropyl)-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
4-methyl-5-(2-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-thiazole
1-(6-aminopyridine-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
6-(1-methyl-1H-imidazol-2-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyridazin-3-amine
N-({7-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
8-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(1H-imidazol-4-yl)-1-[(2S)-oxolan-2-ylmethyl]-1H-imidazole
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine