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[5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)furan-2-yl]methanol
1-[benzyl(methyl)amino]-3-(2-methoxy-5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
[(2,2-dimethyl-1-phenylcyclopropyl)methyl]({[2-(2-methoxyethyl)pyrimidin-5-yl]methyl})methylamine
5-[(dimethylamino)methyl]-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazole-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1H-imidazol-2-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-({[(4,6-dimethylpyrimidin-2-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
(3aS,6aS)-2-[(5-acetylthiophen-3-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-5-methyl-1H-pyrazole-3-carboxamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-2-[4-(4-methylpiperazin-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
methyl 6-{[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]amino}-1,2,3,4-tetrahydroquinoline-1-carboxylate
N-methyl-3-[(3R,4S)-3-[2-(2-methylphenyl)acetamido]-4-(propan-2-yl)pyrrolidin-1-yl]propanamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(1H-indol-2-ylmethyl)(2-methoxyethyl)amine
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}acetamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
1-(2-methoxyphenyl)-4-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
N-(3-fluorophenyl)-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
2-[1-(2,6-difluorobenzenesulfonyl)azetidin-3-yl]pyridine
N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
3-[2-(3-chlorophenyl)-2-hydroxyacetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-[6-chloro-3-(1H-imidazol-2-yl)imidazo[1,2-a]pyridine-2-carbonyl]azocane
N-[2-(1H-indol-1-yl)ethyl]-N-methyloxane-4-carboxamide
2-{2-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
6-(azepan-1-yl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
[1-(1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidin-3-yl)piperidin-4-yl]methanol
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(4-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclopropylmethyl)-5-{[2-(7-methyl-1H-indol-3-yl)ethyl]amino}azepan-2-one
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
2-(3-ethyl-2-imino-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
2-[4-(2-phenoxyethyl)piperazin-1-yl]quinoline
1-(1'-{thieno[3,2-d]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
[3-(2-methoxyethyl)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidin-3-yl]methanol
4-[2-(6-fluoro-2-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-1,4-oxazepan-5-one
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-cyclopropyl-4-hydroxy-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]pyrimidine-5-carboxamide
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-phenylethane-1,2-dione
3-(3-fluorophenyl)-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one
3-fluoro-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
6-methyl-N-[1-(morpholin-4-yl)propan-2-yl]-2-phenylpyrimidin-4-amine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}pyrrolidin-3-ol
(1-{[2-(furan-2-yl)phenyl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
2-methoxy-4-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}benzamide
2-[(3,5-dimethylphenyl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-cyclopropyl-3-{5-[(5-methylfuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[2-(furan-2-yl)-2-hydroxyethyl]-2,3-dimethyl-1H-indole-7-carboxamide
2-methyl-6-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyrimidin-4-ol